Studies on Peptides. LXXIV. Convenient Procedure for the Preparation of Methionine Sulphoxide Derivatives

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概要

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• Sodium perborate can be used for oxidation of N^α-protected Met derivatives to the corresponding (R, S)-sulphoxide. Thus a new derivative, Z(OMe)-Met-(R, S)-sulphoxide was easily prepared in good yield. Sodium metaperiodate was also employed for this purpose.

• 公益社団法人日本薬学会の論文
• 1978-02-25

著者

• 藤井 信孝

  Faculty of Pharmaceutical Sciences, Kyoto University

• 矢島 治明

  Faculty of Pharmaceutical Sciences, Kyoto University

• 佐々木 敬

  Research Institute Daiichi Seiyaku Co. Ltd.

• 船越 奨

  Faculty of Pharmaceutical Sciences

• 佐々木 敬

  Faculty of Pharmaceutical Sciences, Kyoto University

• 入江 寛

  長崎大学薬学部

• 入江 寛

  Faculty Of Pharmaceutical Sciences Kyoto University

• 矢島 治明

  Faculty Of Pharmaceutical Sciences Kyoto University

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