Studies on Peptides. XLVIII. Application of the Trifluoromethanesulphonic Acid Procedure to the Synthesis of Tuftsin
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概要
- 論文の詳細を見る
Trifluoromethanesulphonic acid removed all protecting groups from Z-Thr-Lys (Z)-Pro-Arg (Tos)-OH to give the phagocytosis-stimulating tetrapeptide, H-Thr-Lys-Pro-Arg-OH, named tuftsin. To this synthesis, the 5-chloro-8-quinolyl ester procedure was applied. With this connection, a number of analogous active esters was prepared.
- 社団法人日本薬学会の論文
- 1975-02-25
著者
-
藤井 信孝
Faculty of Pharmaceutical Sciences, Kyoto University
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小川 博
Faculty Of Pharmaceutical Sciences Kyoto University
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