Condensed Heteroaromatic Ring Systems. XXI.Synthesis of Pyrrolo[2,3-d]pyrimidines and pyrrolo[3,2-d]pyrimidines

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概要

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• Pyrrolo[2,3-d]pyrimidines and pyrrolo[3,2-d]pyrimidines were synthesized in high yields by the palladiumcatalyzed reaction of 4-acetylamino-5-bromopyrimidines and 5-acetylamino-4-iodopyrimidines with (Z)-1-ethoxy-2-(tributylstannyl)ethene followed by cyclization under acidic conditions.

• 公益社団法人日本薬学会の論文
• 1993-01-15

著者

• 根東 義則

  Pharmaceutical Institute, Tohoku University

• 坂本 尚夫

  Pharmaceutical Institute, Tohoku University

• 山中 宏

  Pharmaceutical Institute, Tohoku University

• 根東 義則

  Graduate School Of Pharmaceutical Sciences Tohoku University

• 坂本 尚夫

  東北大院薬

• 坂本 尚夫

  Pharmaceutical Institute Tohoku University

• 坂本 尚夫

  東北大学大学院薬学研究科

• 佐藤 千里

  Pharmaceutical Institute, Tohoku University

• 佐藤 千里

  Pharmaceutical Institute Tohoku University

関連論文

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