Condensed Heteroaromatic Ring Systems. XIII. : One-Step Synthesis of 2-Substituted 1-Methylsulfonylindoles from N-(2-Halophenyl)methanesulfonamides

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概要

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• The reaction of N-(2-bromophenyl)-and N-(2-iodophenyl)methanesulfonamide with terminal acetylenes in the presence of dichlorobis(triphenylphosphine)palladium yielded 1-methylsulfonyl-indoles having carbon-functional groups at the 2-position, such as hydroxmethyl, 2-hydroxyethyl, diethoxymethyl, 2-ethoxycarbonylethyl, etc., in one step.

• 公益社団法人日本薬学会の論文
• 1988-04-25

著者

• 根東 義則

  Pharmaceutical Institute, Tohoku University

• 坂本 尚夫

  Pharmaceutical Institute, Tohoku University

• 山中 宏

  Pharmaceutical Institute, Tohoku University

• 根東 義則

  Graduate School Of Pharmaceutical Sciences Tohoku University

• 坂本 尚夫

  東北大院薬

• 坂本 尚夫

  Pharmaceutical Institute Tohoku University

• 坂本 尚夫

  東北大学大学院薬学研究科

• 永野 辰夫

  Pharmaceutical Institute, Tohoku University

• 岩下 茂樹

  Pharmaceutical Institute, Tohoku University

• 岩下 茂樹

  Pharmaceutical Institute Tohoku University

• 永野 辰夫

  Pharmaceutical Institute Tohoku University

関連論文

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