Studies on Pyrimidine Derivatives. XXI. Nucleophilic Substitution of 4-Chloropyrimidines and Related Compounds with Carbanions
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概要
- 論文の詳細を見る
The reaction of 4-chloro-2,6-dimethylpyrimidine 1-oxide (II) with ethyl cyanoacetate and malononitrile under basic conditions gave the expected condensation products, while the reaction of II with methylene ketones failed. On the other hand, 2,6-dimethyl-4-phenylsulfonylpyrimidine (X) smoothyl reacted not only with the above active methyl compounds but also with methylene ketones such as acetone, acetophenone and cyclohexanone.
- 公益社団法人日本薬学会の論文
- 1981-01-25
著者
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小川 茂
Pharmaceutical Institute Tohoku University
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山中 宏
Pharmaceutical Institute, Tohoku University
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今野 昌悦
東北大学薬学部
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今野 昌悦
Pharmaceutical Institute, Tohoku University
関連論文
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