Condensed Heteroaromatic Ring Systems. VIII. : Synthesis of 3-Substituted Isocoumarins from o-Halobenzoic Acid Derivatives
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概要
- 論文の詳細を見る
The hydration of o-ethynylbenzoic acid derivatives, such as ethyl o-ethynylbenzoate, o-ethynylbenzonitrile, and o-ethynylbenzamide, in sulfuric acid in the presence of marcuric sulfate, afforded 3-substituted isocoumarins. The palladium-catalyzed reaction of o-halobenzoic acid derivatives with terminal acetylenes to obstain the starting materials for the cyclization is also described.
- 公益社団法人日本薬学会の論文
- 1986-07-25
著者
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根東 義則
Pharmaceutical Institute, Tohoku University
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山中 宏
Pharmaceutical Institute, Tohoku University
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坂本 尚夫
東北大院薬
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坂本 尚夫
Pharmaceutical Institute Tohoku University
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坂本 尚夫
東北大学大学院薬学研究科
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安中 正幸
Pharmaceutical Institute, Tohoku University
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安中 正幸
Pharmaceutical Institute Tohoku University
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