Reaction of Benzoxazoline-2-thiones with Alkyl Halides

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概要

• 論文の詳細を見る

• The effect of the solvent on the reaction of benzoxazoline-2-thiones with alkyl halides was studied. The reaction of 1 with alkyl halides and potassium carbonate in dimethylformamide (DMF) gave the corresponding 2-alkylthiobenzoxazoles (2), but the same reaction gave 2-methoxybenzoxazoles (4a) when methanol was used in place of DMF as the solvent. On the other hand, the reaction of 1,methyl iodide, alcohol, and sodium hydride in tetrahydrofuran (THF) gave 2-[N-(dialkoxymethylene) amino] phenols (5).

• 社団法人日本薬学会の論文
• 1983-02-25

著者

• 竹内 靖雄

  岡山大学薬学部

• 竹内 靖雄

  Faculty of Pharmaceutical Sciences, Okayama University

• 橋垣 国子

  Faculty of Pharmaceutical Sciences, Okayama University

• 大和 正利

  Faculty of Science, Okayama University of Science

• 広田 喬

  Faculty of Pharmaceutical Sciences, University

• 廣田 喬

  Faculty Of Pharmaceutical Sciences Okayama University

• 大和 正利

  Faculty Of Pharmaceutical Sciences Okayama University

• 竹内 靖夫

  Faculty Of Pharmaceutical Sciences Okayama University:cancer Chemotherapy Center

• 広田 喬

  岡山大学 薬

• 橋垣 国子

  Faculty Of Pharmaceutical Sciences Okayama University

• 橋垣 國子

  Faculty Of Pharmaceutical Sciences Okayama University

• 広田 喬

  Faculty Of Pharmaceutical Sciences Okayama University

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