Polycyclic N-Hetero Compounds. II, Synthesis of 11,13,15-Triazasteroidal Skeleton
スポンサーリンク
概要
- 論文の詳細を見る
Heating of 2-cyano-1-tetralones (I) with formamide and phosphoryl chloride afforded 4-amino-5,6-dihydrobenzo [h] quinazolines (II). 4-(2-Hydroxyethylamino)-5,6-dihydrobenzo [h] quinazolines (III) were obtained from II with ethylene chlorohydrin, and gave 1,2,4,5-tetrahydrobenz [h] imidazo [1,2-c] quinazolines (V), i.e., 11,13,15-triazasteroid compounds, on treatment with sodium carbonate after refluxing with phosphorus tribromide.
- 社団法人日本薬学会の論文
- 1974-07-25
著者
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原 秀樹
Faculty Of Pharmaceutical Sciences Medical School Okayama University
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大森 晋爾
Faculty of Pharmaceutical Sciences, Medical School, Okayama University
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廣田 喬
Faculty Of Pharmaceutical Sciences Okayama University
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大森 晋爾
Faculty Of Pharmaceutical Sciences Okayama University
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広田 喬
岡山大学 薬
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