Polycyclic N-Hetero Compounds. XI. The Modified Vilsmeier Reaction of 4-Alkylpyrimidines

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概要

• 論文の詳細を見る

• Reactions of 4-alkylpyrimidines with formamide in the presence of phosphoryl chloride (called the modified Vilsmeier reaction) were described. 4-Methylpyrimidine derivatives (I, III) gave 4-pyrimidinylpyrimidines (II, IV) respectively but 4-methylenepyrimidine derivatives (V, VII) afforded 5-hydroxy-6-[4-(5-methylpyrimidinyl)]-2,4-diaza-2-heptenal (VI) or bis (5,6,7,8-tetrahydro-8-quinazolinylidenemethyl) amine (VIII) and 8-formylaminomethinyl-5,6,7,8-tetrahydroquinazoline (IX).

• 公益社団法人日本薬学会の論文
• 1976-07-25

著者

• 大和 正利

  Faculty of Science, Okayama University of Science

• 小山 鷹二

  Faculty of Pharmaceutical Sciences, Medical School, Okayama University

• 大森 晋爾

  Faculty of Pharmaceutical Sciences, Medical School, Okayama University

• 廣田 喬

  Faculty Of Pharmaceutical Sciences Okayama University

• 大森 晋爾

  Faculty Of Pharmaceutical Sciences Okayama University

• 大和 正利

  Faculty Of Pharmaceutical Sciences Okayama University

• 佐藤 美子

  Faculty Of Pharmaceutical Sciences Medical School Okayama University

• 馬生 千鶴子

  Faculty of Pharmaceutical Sciences, Medical School, Okayama University

• 渡辺 靖子

  Faculty of Pharmaceutical Sciences, Medical School, Okayama University

• 渡辺 靖子

  Faculty Of Pharmaceutical Sciences Medical School Okayama University

• 馬生 千鶴子

  Faculty Of Pharmaceutical Sciences Okayma University

• 広田 喬

  岡山大学 薬

• 小山 鷹二

  Faculty Of Pharmaceutical Sciences Okayama University

• 北内 陽子

  Faculty of Pharmaceutical Sciences, Medical School, Okayama University

• 馬生 千鶴子

  Faculty Of Pharmaceutical Sciences Okayama University

• 北内 陽子

  Faculty Of Pharmaceutical Sciences Medical School Okayama University

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