Synthesis of a Griseofulvin Analogue

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概要

• 論文の詳細を見る

• Ring contraction of 6-ethoxycarbonyl-4,5,7-trihydroxycoumarin (7) to a 3(2H)-benzofuranone (13) was achieved. Compound 13 was utilized in a synthesis of a griseofulvin analogue (1b) with an ethoxycarbonyl group at the 5 position. However, 1b was found to be inactive in a test of fungicidal activity.

• 公益社団法人日本薬学会の論文
• 1986-01-25

著者

• 大和 正利

  Faculty of Science, Okayama University of Science

• 大和 正利

  Faculty Of Pharmaceutical Sciences Okayama University

• 大和 正利

  Faculty Of Science Okayama University Of Science

• 吉田 浩一

  Faculty Of Pharmaceutical Sciences Okayama University

• 池沢 喜三雄

  Faculty of Pharmaceutical Sciences, University of Okayama

• 小橋 芳枝

  Faculty of Pharmaceutical Sciences, University of Okayama

• 小橋 芳枝

  Faculty Of Pharmaceutical Sciences University Of Okayama

• 池沢 喜三雄

  Faculty Of Pharmaceutical Sciences University Of Okayama

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