Polycyclic N-Hetero Compounds. XVII. Reactions of Heterocyclic Active Methyl Group with Formamide or Trisformylaminomethane

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概要

• 論文の詳細を見る

• Pyrimidine formation from active methyl group on heterocycles is described. 2-Methyl-pyridine (I), -quinoline (III), -pyrazine (IX), -benzothiazole (XX), 2,4-dimethylquinoline (VII), and-thiazole (XIII) were successful in pyrimidine formation. 2-Methylimidazole (XI), -benzimidazole (XV), -benzoxazole (XVI), and 2,4-dimethyloxazole (XII) were unsuccessful. Compound (III) gave pyrazine (V) and pyridine (VI) derivatives and pyridine formation occurred also in XX.

• 公益社団法人日本薬学会の論文
• 1977-11-25

著者

• 大和 正利

  Faculty of Science, Okayama University of Science

• 小山 鷹二

  Faculty of Pharmaceutical Sciences, Medical School, Okayama University

• 廣田 喬

  Faculty Of Pharmaceutical Sciences Okayama University

• 大和 正利

  Faculty Of Pharmaceutical Sciences Okayama University

• 佐々木 健二

  Faculty Of Pharmaceutical Sciences Okayama University

• 馬生 千鶴子

  Faculty of Pharmaceutical Sciences, Medical School, Okayama University

• 難波 哲人

  Faculty of Pharmaceutical Sciences, Okayama University

• 馬生 千鶴子

  Faculty Of Pharmaceutical Sciences Okayma University

• 難波 哲人

  Faculty Of Pharmaceutical Sciences Okayama University

• 広田 喬

  岡山大学 薬

• 小山 鷹二

  Faculty Of Pharmaceutical Sciences Okayama University

• 馬生 千鶴子

  Faculty Of Pharmaceutical Sciences Okayama University

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