Polycyclic N-Hetero Compounds. X. Reactions of 1,3-Cyclohexanedione and Its Dimer with Formamide or Trisformylaminomethane

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概要

• 論文の詳細を見る

• Condensation of 1,3-cyclohexanedione (I) with formamide gave 9,10-dihydro-1,3,5,7-tetraazaphenanthrene (II), 1,2,3,4,5,6,7,8,9,10-decahydro-11,13-diazabenzo [g] chrysene-1,-5-dione (III), 1,2,5,6-tetrahydro-3,7,9,11,13-pentaazadibenzophenanthrene (IV), and 7,8,13,14-tetrahydro-2,4,6,10,12-pentaazabenzo [c] chrysene (V). Dehydrogenation of II with sulfur gave 1,3,5,7-tetraazaphenanthrene (VI). To make sure the formation mechanism of IV and V, dimer of I (enol form of VII') was heated with formamide or trisformyl-aminomethane and the formation of IV and V were confirmed.

• 公益社団法人日本薬学会の論文
• 1976-04-25

著者

• 大和 正利

  Faculty of Science, Okayama University of Science

• 小山 鷹二

  Faculty of Pharmaceutical Sciences, Medical School, Okayama University

• 大森 晋爾

  Faculty of Pharmaceutical Sciences, Medical School, Okayama University

• 廣田 喬

  Faculty Of Pharmaceutical Sciences Okayama University

• 大森 晋爾

  Faculty Of Pharmaceutical Sciences Okayama University

• 大和 正利

  Faculty Of Pharmaceutical Sciences Okayama University

• 前田 純

  Faculty Of Pharmaceutical Sciences Medical School Okayama University

• 広田 喬

  岡山大学 薬

• 小山 鷹二

  Faculty Of Pharmaceutical Sciences Okayama University

• 福岡 純男

  Faculty of Pharmaceutical Sciences, Medical School, Okayama University

• 福岡 純男

  Faculty Of Pharmaceutical Sciences Medical School Okayama University

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