Benzylcarbonyl化合物とFormamideとの反応(第9報)α-Acyl-5,6,7,8-tetrahydro-2-naphthylacetonitrileとの反応

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概要

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• Treatment of α-formyl-(IIa) and α-acetyl-5,6,7,8-tetrahydronaphthyl-2-acetonitrile (IIb) with formamide and phosphoryl chloride respectivily gave 4-amino-(IIIa) and 4-amino-6-methyl-5-(5,6,7,8-tetrahydro-2-naphthyl) pyrimidine (IIIc). The same treatment of the benzoyl derivative (IIc) gave IIIa and benzamide (IV).

• 公益社団法人日本薬学会の論文
• 1973-11-25

著者

• 廣田 喬

  Faculty Of Pharmaceutical Sciences Okayama University

• 小山 鷹二

  岡山大学医学部附属病院薬剤部

• 大和 正利

  Faculty Of Pharmaceutical Sciences Okayama University

• 廣田 喬

  岡山大学医学部薬学科

• 大和 正利

  岡山大学医学部薬学科

• 構木 信也

  吉富製薬株式会社

• 小山 鷹二

  岡山大学医学部付属病院薬剤部

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