Polycyclic N-Hetero Compounds. XIII. Reactions of Pyridine N-Oxides with Formamide

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概要

• 論文の詳細を見る

• Reactions of pyridine (I, IV, X, XIII) or condensed pyridine (VII, XVI, XVIII) N-oxides with formamide were described. Although pyrimidinyl cyclization of active methyl group was unsuccessful, introduction of carbamoyl group at pyridine ring carbon adjacent to nitrogen atom was successful, i. e., 6-methylpyridine-2-(II), 4-methylpyridine-2-(V), 4-methylquinoline-2-(VIII), 5-methylpyridine-2-(XI), pyridine-2-(XIV), quinoline-2-(XVII), and isoquinoline-1-(XIX) carboxyamides were obtained.

• 公益社団法人日本薬学会の論文
• 1977-05-25

著者

• 大和 正利

  Faculty of Science, Okayama University of Science

• 小山 鷹二

  Faculty of Pharmaceutical Sciences, Medical School, Okayama University

• 大森 晋爾

  Faculty of Pharmaceutical Sciences, Medical School, Okayama University

• 廣田 喬

  Faculty Of Pharmaceutical Sciences Okayama University

• 大森 晋爾

  Faculty Of Pharmaceutical Sciences Okayama University

• 大和 正利

  Faculty Of Pharmaceutical Sciences Okayama University

• 難波 哲人

  Faculty of Pharmaceutical Sciences, Okayama University

• 難波 哲人

  Faculty Of Pharmaceutical Sciences Okayama University

• 広田 喬

  岡山大学 薬

• 小山 鷹二

  Faculty Of Pharmaceutical Sciences Okayama University

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