1,3,10-Triazaphenanthreneの合成(第1報)

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概要

• 論文の詳細を見る

• 4-Amino-5-(3,5-dimethoxyphenyl) pyrimidine (II) and 4-amino-5-(3-methoxyphenyl)-pyrimidine (VI) were acetylated to 4-acetamido-5-(3,5-dimethoxyphenyl) pyrimidine (III) and 4-acetamido-5-(3-methoxyphenyl) pyrimidine (VII). III and VII gave respectively gave 6,8-dimethoxy-9-methyl-1,3,10-triazaphenanthrene (IV)+(II) and 6-methoxy-9-methyl-1,3,10-triazaphenanthrene (VIII)+(VI) by the Bischler-Napieralski cyclization with polyphosphoric acid. This is a novel synthetic method for 1,3,10-triazaphenanthrene derivarives.

• 公益社団法人日本薬学会の論文
• 1973-03-25

著者

• 廣田 喬

  Faculty Of Pharmaceutical Sciences Okayama University

• 小山 鷹二

  岡山大学医学部附属病院薬剤部

• 大和 正利

  Faculty Of Pharmaceutical Sciences Okayama University

• 廣田 喬

  岡山大学医学部薬学科

• 大和 正利

  岡山大学医学部薬学科

• 太田 直角

  熊本大学薬学部

• 小山 鷹二

  岡山大学医学部付属病院薬剤部

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