Studies on Ketene and Its Derivatives. XCV. Reaction of Diketene with Acyl Azides

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概要

• 論文の詳細を見る

• Photolysis of acyl azides (1,10) in diketene was investigated. Irradiation of a mixture of benzoyl azide (1a) and diketene in dichloromethane gave 1-benzoyl-4-hydroxy-3-pyrrolin-2-one (2a) in 17% yield. Similarly, reaction of diketene with p-anisoyl azide (1b), p-toluoyl azide (1c), p-chlorobenzoyl azide (1d) and ethyl azidoformate (10) gave the corresponding pyrrolinones (2b, 2c, 2d, and 11) in 7-22% yields.

• 社団法人日本薬学会の論文
• 1979-05-25

著者

• 佐藤 雅之

  静岡県立大学薬学部

• 鈴木 雄二

  Hoshi College Of Pharmacy

• 佐藤 雅之

  Pharmaceutical Institute, Tohoku University

• 加藤 鉄三

  東北大学 薬

• 加藤 鉄三

  Pharmaceutical Institute Tohoku University

• 鈴木 雄二

  Pharmaceutical Institute, Tohoku University

• 加藤 鉄三

  Pharmaceutical Institute. Tohoku University

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