Synthesis of a Nitrogen Analogue of Salacinol and Its α-Glucosidase Inhibitory Activity
スポンサーリンク
概要
- 論文の詳細を見る
A nitrogen analogue 4 of the naturally occurring sulfonium ion salacinol (1), a potent α-glucosidase inhibitor isolated from the Ayruvedic medicine Salacia reticulata, was synthesized and its inhibitory activity against α-glucosidase tested. Substitution of the sulfur atom in 1 with a nitrogen reduced the activity considerably. The solid-state stereostructure of the related compound (5) was determined on the basis of single crystal X-ray measurement.
- 社団法人日本薬学会の論文
- 2001-11-01
著者
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MATSUDA Hisashi
Kyoto Pharmaceutical University
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YOSHIKAWA Masayuki
Kyoto Pharmaceutical University
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吉川 雅之
Kyoto Pharmaceutical Univ.
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Muraoka Osamu
Pharmaceutical Research and Technology Institute, Kinki University
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Muraoka Osamu
Pharmaceutical Research And Technology Institute Kinki University
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Muraoka Osamu
近畿大学薬学総合研究所
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Muraoka Osamu
School of Pharmacy, Kinki University
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Tanabe Genzoh
School of Pharmacy, Kinki University
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Yoshikai Kazuya
School of Pharmacy, Kinki University
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Minematsu Toshie
School of Pharmacy, Kinki University
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YING Shao
School of Pharmaceutical Sciences, Kinki University
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MATSUURA Yoshiharu
School of Pharmaceutical Sciences, Kinki University
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YAMADA Eriko
School of Pharmaceutical Sciences, Kinki University
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Tanabe Genzoh
近畿大学 薬
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Ying Shao
School Of Pharmaceutical Sciences Kinki University
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Yamada Eriko
Pharmaceutical Research And Technology Institute Kinki University
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Yamada E
Kinki Univ. Osaka Jpn
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Tanabe Genzoh
School Of Pharmacy Kinki University
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Tanabe Genzoh
School Of Pharmaceutical Sciences Kinki University
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Muraoka Osamu
School Of Pharmaceutical Sciences Kinki University
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Yamazaki M
School Of Pharmaceutical Sciences Kinki University
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Tanabe Genzoh
School Of Pharmacy Kinki Univ.
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Yoshikai Kazuya
School Of Pharmacy Kinki University
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Minematsu T
School Of Pharmaceutical Sciences Kinki University
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Minematsu Toshie
School Of Pharmaceutical Sciences Kinki University
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Minematsu Toshie
School Of Pharmacy Kinki University
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MATSUDA HISASHI
Kyoto College of Pharmacy
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