Binding Selectivity of Conformationally Restricted Analogues of (-)-Indolactam-V to the C1 Domains of Protein Kinase C Isozymes(Organic Chemistry)
スポンサーリンク
概要
- 論文の詳細を見る
Two conformationally restricted analogues of (-)-indolactam-V (1) (cis and trans amides) were examined for their binding selectivity to the synthetic C1 peptides of all protein kinase C (PKC) isozymes. Although the binding constants of the cis amide-restricted analogue (2) were equal to those of 1, the trans amide-restricted analogue (3) bound significantly only to the novel PKC (δ, ε, η, θ) isozymes.
- 社団法人日本農芸化学会の論文
- 2002-07-23
著者
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OHIGASHI Hajime
Division of Food Science and Biotechnology, Graduate School of Agriculture, Kyoto University
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Ohigashi H
Department Of Surgery Osaka Medical Center For Cancer And Cardiovascular Diseases
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Ohigashi Hiroaki
Department Of Surgery The Center For Adult Diseases
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入江 一浩
京都大学農学部
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入江 一浩
京都大学 食品工学
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入江 一浩
京都大学 農
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入江 一浩
京都大学大学院農学研究科食品生物科学
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Nakamura Yoshimasa
Division Of Applied Life Sciences Graduate School Of Agriculture Kyoto University
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Nakamura Y
Division Of Applied Life Sciences Graduate School Of Agriculture Kyoto University
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Ohigashi H
Graduate School Of Agriculture Kyoto University
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Ohigashi H
Division Of Applied Life Sciences Graduate School Of Agriculture Kyoto University
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Nakagawa Y
Graduate School Of Agriculture Kyoto University
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Nakagawa Yu
Graduate School Of Agriculture Kyoto University
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Nakagawa Yasue
Department Of Food Faculty Of Home Economics Jissen Women's University
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Ohigashi Hajime
Division Of Applied Life Sciences Graduate School Of Agriculture Kyoto University
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IRIE KAZUHIRO
Division of Food Science and Biotechnology, Graduate School of Agriculture, Kyoto University
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NAKAGAWA Yu
Division of Applied Life Sciences, Graduate School of Agriculture, Kyoto University
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Masuda Akiko
Division Of Food Science And Biotechnology Graduate School Of Agriculture Kyoto University
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Irie Kazuhiro
Division Of Food Science And Biotechnology Graduate School Of Agriculture Kyoto University
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入江 一浩
Division Of Food Science And Biotechnology Graduate School Of Agriculture Kyoto University
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Nakagawa Yu
Division Of Food Science And Biotechnology Graduate School Of Agriculture Kyoto University
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