Synthesis and Biological Activities of Indolactone-V, the Lactone Analogue of the Tumor Promoter (-)-Indolactam-V
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概要
- 論文の詳細を見る
The tumor promoter (-)-indolactam-V (1) exists in two stable conformers (twist and sofa) due to isomerization of the amide group. Indolactone-V (2), the lactone analogue of 1, has been synthesized to investigate the effects of the amide group on its conformation and biological actirities. Indolactone-V (2) existed only as the inactive sofa-like conformer, indicating that the amide group of 1 plays a critical role in formation of the active twist conformation.
- 社団法人日本農芸化学会の論文
- 1997-08-23
著者
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OHIGASHI Hajime
Division of Food Science and Biotechnology, Graduate School of Agriculture, Kyoto University
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Ohigashi H
Department Of Surgery Osaka Medical Center For Cancer And Cardiovascular Diseases
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Ohigashi Hiroaki
Department Of Surgery The Center For Adult Diseases
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入江 一浩
京都大学農学部
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入江 一浩
京都大学 食品工学
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入江 一浩
京都大学 農
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入江 一浩
京都大学大学院農学研究科食品生物科学
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Nakamura Yoshimasa
Division Of Applied Life Sciences Graduate School Of Agriculture Kyoto University
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Nakamura Y
Division Of Applied Life Sciences Graduate School Of Agriculture Kyoto University
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Ohigashi H
Graduate School Of Agriculture Kyoto University
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Ohigashi H
Division Of Applied Life Sciences Graduate School Of Agriculture Kyoto University
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HAYASHI Hideo
Deparment of Applied Biological Chemistry, College of Agriculture, Osaka Prefecture University
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Nakagawa Y
Graduate School Of Agriculture Kyoto University
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Nakagawa Yu
Graduate School Of Agriculture Kyoto University
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Hayashi H
Osaka Prefecture Univ. Osaka Jpn
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Nakagawa Yasue
Department Of Food Faculty Of Home Economics Jissen Women's University
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Ohigashi Hajime
Division Of Applied Life Sciences Graduate School Of Agriculture Kyoto University
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IRIE KAZUHIRO
Division of Food Science and Biotechnology, Graduate School of Agriculture, Kyoto University
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NAKAGAWA Yu
Division of Applied Life Sciences, Graduate School of Agriculture, Kyoto University
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Irie Kazuhiro
Division Of Food Science And Biotechnology Graduate School Of Agriculture Kyoto University
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入江 一浩
Division Of Food Science And Biotechnology Graduate School Of Agriculture Kyoto University
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Nakagawa Yu
Division Of Food Science And Biotechnology Graduate School Of Agriculture Kyoto University
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