Phytogrowth-Inhibitory and Antimicrobial Activities of 3,4'-Dihydroxy-α, β-diethylstilbene, the Isomer of Diethylstilbestrol

スポンサーリンク

概要

• 論文の詳細を見る

• 3,4'-Dihydroxy-α, β-diethylstilbene (I), like diethylstilbestrol (II), showed phytogrowth-inhibitory and antimicrobial activities. First, compound I showed strong growth-inhibitory activity against the roots of two kinds of plants. The inhibitory activity of I was almost equal to that of sodium 2,4-dichlorophenoxyacetate used as a positive control. The phytogrowth-inhibitory activity of I was much higher than that of II. Next, unlike II, I had broad antifungal spectrum against pathogenic fungi. Compound I showed antifungal activity against six kinds of Fusarium oxysporum sp. This compound also had antibacterial activity against pathogenic and plant-pathogenic bacteria. These antibacterial activities of I were as high as those of II, the isomer of I. It should be emphasized that by shifting one of the phenolic hydroxyl groups of II to meta-position, phytogrowth-inhibitory activity was largely increased, while antimicrobial activity was unchanged.

• 社団法人日本薬学会の論文
• 1991-01-25

著者

• 竹村 庄司

  Faculty Of Pharmaceutical Sciences Kinki University

• 稲森 善彦

  Osaka University of Pharmaceutical Sciences

• 辻坊 裕

  Osaka University of Pharmaceutical Sciences

• 小山 智子

  Osaka University Of Pharmaceutical Sciences

• 小川 雅史

  Osaka University Of Pharmaceutical Sciences

• 三木 康義

  Faculty of Pharmaceutical Sciences, Kinki University

• 西口 一基

  Osaka University of Pharmaceutical Sciences

• 辻坊 裕

  大阪薬大

• 三木 康義

  Faculty Of Pharmaceutical Sciences Kinki University

• 三木 康義

  近畿大学 薬学部

• 竹村 庄司

  Faculty of Pharmaceutical Sciences, Kinki University

関連論文

• Antibacterial Activity of Two Chalcones, Xanthoangelol and 4-Hydroxyderricin, Isolated from the Root of Angelica keiskei KOIDZUMI
• 藻類およびコケ培養細胞に対する rhodanine と 2(5H)-thiophenone の効果
• Phytogrowth-Inhibitory Activities of 2-Thiophenecarboxylic Acid and Its Related Compounds
• Phytogrowth-Inhibitory Activities of Sulfur-Containing Compounds. II.The Inhibitory Activities of Thiosalicylic Acid and Dihydro-2(3H)-thiophenone-Related Compounds on Plant Growth
• Phytogrowth-Inhibitory Activity of Sulphur-Containing Compounds. I. Inhibitory Activities of Thiazolidine Derivatives on Plant Growth
• Relationship between Structure and Phytogrowth-Inhibitory Activity of 2,5-Dihydroxy-1,4-dithiane-Related Compounds
• Pharmacokinetics of Cyproheptadine and Its Metabolites in Rats
• Structure-Activity Relationship of 3,3'-Dihydroxy-α, β-diethyldiphenylethane and Its Related Compounds
• Inhibitory Effects of 3,3', 4,5'-Tetrahydroxystilbene and 3,3', 4,5'-Tetrahydroxybibenzyl, the Constituents of Cassia garrettiana on Antigen-Induced Histamine Release in Vitro
• THE INHIBITORY EFFECT OF 3,3', 4,5'-TETRAHYDROXYSTILBENE, A CONSTITUENT OF CASSIA GARRETTIANA, ON ANTI-IgE-INDUCED HISTAMINE RELEASE FROM HUMAN BASOPHILS IN VITRO
• Phytogrowth-Inhibitory and Antimicrobial Activities of 3,4'-Dihydroxy-α, β-diethylstilbene, the Isomer of Diethylstilbestrol
• Hypotensive Effects on Spontaneously Hypertensive Rats and Antifungal Activity on Various Species of Fusarium oxysporum of Diethylstilbestrol-Related Compounds
• The Hypotensive Effect and Antifungal Activity of 3,3'-Dihydroxy-α, β-diethyldiphenylethane
• Antifungal Activity against Plant-Pathogenic Fungi and Phytogrowth-Inhibitory Activity of 3,3'-Dihydroxy-α, β-diethyldiphenylethane
• Biological Actibities of Hexesterol
• THE ICHTHYOTOXICITY AND CORONARY VASODILATOR ACTION OF 3,3'-DIHYDROXY-α,β-DIETHYLSTILBENE(Communications to the Editor)
• The Biological Activities of Podophyllotoxin Compounds
• The Biological Activities of Diethylstilbestrol and Its Derivatives
• THE ICHTHYOTOXICITY AND CORONARY VASODILATOR ACTION OF DIETHYLSTILBESTROL
• Novel Hypotensive Peptides from the Body of Elaphe climacophora
• Antimicrobial Activity on Plant-Pathogenic Microorganisms and Phytogrowth-Inhibitory Activity of Streptothricin Antibiotics, Racemomycin-A and -C
• モノテルペンの生物学的特性 モノテルペンのラットに対する血圧降下作用と植物病原真菌に対する抗真菌効果
• Phytogrowth-Inhibitory Activities of Tropolone and Hinokitiol
• 写真処理廃液中に含まれるEDTA鉄キレート分解菌株A-1の特性
• Determination of β-Lactam Antibiotics in Water by Fluorescence Quenching of Mercurochrome, and Application for Simple Investigation of Potency
• Study on Conformations-Biological Activities Relationships for Podophyllotoxin Analogues Based on Crystal Structure of Deoxypodophyllotoxin (Anthricin)
• Studies on the Constituents of the Water Extract of the Root of Mulberry Tree (Morus bombycis KOIDZ)
• Synthesis and Bioactivity of Propranolol Analogues with a Rigid Skeleton. I
• Synthesis and Selective Activity of Cholinergic Agents with Rigid Skeletons. IV
• Synthesis and Selective Activity of Cholinergic Agents with Rigid Skeletons. III
• Synthesis and Selective Activity of Cholinergic Agents with Rigid Skeletons. II
• 降圧性コリン作働薬を目的とした合成(2)(II 予防および治療)(A 基礎的研究)
• 降圧性コリン作働薬を目的とした合成(A 基礎的研究)(II 予防および治療)
• Synthesis and Selective Activity of Cholinergic Agents with Rigid Skeletons. I
• The Biological Actions of Deoxypodophyllotoxin (Anthricin). I. Physiological Activities and Conformational Analysis of Deoxypodophyllotoxin
• Cytotoxic Effect of Hinokitiol and Tropolone on the Growth of Mammalian Cells and on Blastogenesis of Mouse Splenic T Cells
• Benzoylthiocholine Derivatives as Substrates for Pseudocholinesterase : Synthesis and Application(Analytical,Chemical)
• Isolation of Cytotoxic Substance, Kalafungin from an Alkalophilic Actinomycete, Nocardiopsis dassonvillei subsp. presina
• ベンズヒドリル誘導体の研究(第2報)N, N-ジアルキルグリシルベンズヒドリルアミド誘導体の合成と生物活性
• Effects of 3,3'-dihydroxy-α, β-diethylstilbene and 3,3', 4,5'-Tetrahydroxystilbene on Microtubule Assembly in Vitro, Aneuploidy Induction, and Cellular Microtubule and Actin Networks
• Toxicological Approaches to Streptothricin Antibiotics. IV. Toxicity of Streptothricin Antibiotics to the Blood
• Reaction of N-Halosulfonamide. IV. A Cleavage Reaction of Ether with N, N-Dihalobenzenesulfonamide. (1).
• Reaction of N-Halosulfonamide. III. Reaction of N, N-Dibromobenzenesulfonamide with Cyclopentene.
• Reaction of DL-trans-and DL-cis-2-Halo-1-benzenesulfonamidocyclohexanes. Formation and the Reaction of N-Benzenesulfonylcyclohexenimine.
• Reaction of N-Halosulfonamide. II. Reaction of N, N-Dihalobenzenesulfonamide with Cyclohexene. (2).
• Reaction of N-Halosulfonamide. I. Reaction of N, N-Dihalobenzenesulfonamide with Cyclohexene. (1).
• Reaction of N, N-Dihalobenzenesulfonamide with Cyclohexene. Formation of DL-trans-and DL-cis-2-Halo-1-benzenesulfonamidocyclohexanes
• Changes of Tissue Histopathology and Uric Acid Excretion in Silkworm Larvae Intoxicated with Deoxypodophyllotoxin and Racemomycin-D, and during Starvation
• Mechanisms of Inhibitory Action of Racemomycin-D on Plant Growth
• The Biological Activities of 3,4-O-Isopropylidene-3,3'4,5'-tetrahydroxystilbene
• Mechanisms of Insecticidal Action of Deoxypodophyllotoxin (Anthricin). II. Histopathological Studies on Tissues of Silkworm Larvae Intoxicated by Deoxypodophyllotoxin
• THE ANTIFUNGAL ACTIVITY OF STILBENE DERIVATIVE
• Physiological Activities of 3,3', 4,5'-Tetrahydroxystilbene Isolated from the Heartwood of Cassia garrettiana CRAIB.
• The Mechanisms of Delayed Insecticidal Action of Streptothricin Antibiotics. I. Toxic Symptoms and Distribution of Racemomycin-D into the Tissues of the 5th Instar Larvae of Silkworm, Bombyx mori LINNE
• The Mechanisms of Delayed Insecticidal Action of Streptothricin Antibiotics. II. Effect of Racemomycin-D on Excretion Function of the 5th Instar Larvae of Silkworm, Bombyx mori LINNE
• Insecticidal Activity of Streptothricin Antibiotics
• Reaction of 2-Methyl-4-phenyl-2,3-dihydro-1H-pyrazolo[2,3,4-de][1,5]-naphthyridine 2-Oxides with Acetic Anhydrides : Polonovski Reaction versus Mesomeric Betaine Formation
• Reaction of N-Haloamide. XIX. Reaction of Acetals with N, N-Dibromobenzenesulfonamide
• Reaction of N-Haloamide. XVIII. Oxidation of Ether to Ester with N-Haloamide
• Reaction of N-Haloamide. XV. Reaction of Tetrahydrofuran with N, N-Dibromobenzenesulfonamide. (2). Kinetics and Mechanism
• Kinetic Studies of the Reaction of Tetrahydrofuran with N-Haloamide under Irradiation
• Steroids from Cucumis Melo L. var. Makuwa MAKINO and Cucumis sativus L.
• Reaction of N-Haloamide. VIII. Reactions of N-Bromobenzenesulfonamides or Bromine with Benzylamines
• Biological Activities of Racemomycin-B, β-Lysine Rich Streptothricin Antibiotic, the Main Component of Streptomyces lavendulae OP-2
• Phytogrowth-Inhibitory and Antibacterial Activities of 2,5-Dihydroxy-1,4-dithiane and Its Derivatives
• EFFECT OF 3,3'-DIHYDROXY-α, β-DIETHYLDIPHENYLETHANE ON CORONARY AND MESENTERIC ARTERIES ISOLATED FROM GUINEA-PIGS
• Studies on Benzhydryl Derivatives. IV. Synthesis and Anti-inflammatory Activity of 2-O-(Diphenylacetyl)salicylic Acids
• ベンズヒドリル誘導体の研究(第3報)ジフェニルアセチルアミノ酸の合成と培養腫瘍細胞におよぼす影響
• 降圧性を目的とした芳香族オキシカルボン酸誘導体の合成(1)(II 予防および治療)(A 基礎的研究)
• 降圧剤を目的としたBenzhydrylidene Guanidine類の合成と活性(II 予防および治療)(A 基礎的研究)
• コリン作働薬の分子座標解析法による構造-活性相関(A 基礎的研究)(II 予防および治療)
• アミノ酸誘導体と生物活性(第2報)フェニルアラニンから2-アミノ-1-インダノール誘導体の合成
• Stability of Enzyme Preparations on Radiosterilization
• Biosynthesis of Streptothricin Antibiotics. III. Incorporation of D-Glucosamine into D-Gulosamine Moiety of Racemomycin-A
• Reaction of N-Haloamide. XXVIII. Preparation of N, N-Dibromourethan and Reactions of N, N-Dihaloamides with Styrene and 1,2-Dihydronaphthalenes
• Reaction of N-Haloamide. XXVII. Reaction of N, N-Dihaloamides with Dienes
• Reaction of N-Haloamide. XXV. Addition Reaction of N, N-Di-bromobenzenesulfonamide with Asymmetric Olefins and α, β-Unsaturated Carboxylic Acid Esters
• Reaction of N-Haloamide. XXIV. N, N-Dibromo-o-carbomethoxybenzene-sulfonamide as a Reagent for the Preparation of β-Substituted Amines from Olefins
• Reaction of N-Haloamide. XXI. Addition Reaction of N, N-Dibromo-benzylsulfonamide with Olefines and Reduction of the Adducts and Their Derivatives
• Reaction of N-Haloamide. XX. Bromo-formyloxylation of α, β-Unsaturated Esters with N, N-Dibromobenzenesulfonamide and Formic Acid
• Reaction of N-Haloamide. XVI. Reaction of N, N-Dichlorophenylacetamide with Aliphatic Secondary Amines
• Reaction of N-Haloamide. XIV. Reaction of N, N-Dichlorophenylacetamide with Cyclohexene
• Reaction of N-Haloamide. XVII. Bromo-formyloxylation of Olefins with N, N-Dibromobenzenesulfonamide and Formic Acid
• Reaction of N-Haloamide. XIII. The Coupled Reaction of N, N-Dibromobenzenesulfonamide and Formamide or Dimethylformamide with Cyclohexene
• Reaction of N-Haloamide. XI. Reaction of N, N-Dichlorobenzenesulfonamide and N, N-Dichlorobenzamide with Dihydropyran
• Reaction of N-Haloamide. X. Reaction of N, N-Dichlorobenzamide with Cyclohexene
• Studies on Benzhydryl Derivatives. I. Synthesis and Anti-Inflammatory Activity
• Chemical Studies on Antibiotics produced by Actinomycetes. VII. Racemomycin. (4). On Racemomycin-O (i)
• Hypotensive Compounds Isolated from Alcohol Extract of the Unossified Horn of Cervus elaphus L. var. xanthopygus MILNE-EDWARG (Rokujo). I. Isolation of Lysophosphatidyl Choline as a Hypotensive Principle and Structure-Activity Study of Related Compounds(P
• CHEMICAL STRUCTURE OF A NEW METABOLITE ISOLATED FROM THE MYCELIUM OF ASPERGILLUS TERREUS VAR. AUREUS
• Mechanism of Insecticidal Action of Deoxypodophyllotoxin(Anthricin). III. : The Mode of Delayed Insecticidal Action of Deoxypodophyllotoxin
• The Mechanisms of Delayed Insecticidal Action of Streptothricin Antibiotics. III. The Mode of Delayed Insecticidal Action of Racemomycin-A(Biological)
• Isomerization between trans-2-Benzenesulfonamido-3-bromotetrahydropyran and Its Isomer
• Reaction of N-Halosulfonamide. VI. Reaction of N-Bromobenzenesulfonamides with Dihydropyran. (2)
• Reaction of N-Halosulfonamide. V. Reaction of N, N-Dibromobenzenesulfonamide with Dihydropyran. (1)
• (250) トマトでのTMVの増殖に対するサルチル酸およびアントラニル酸のベンズヒドリル誘導体の影響 (昭和55年度日本植物病理学会大会講演要旨)
• Reaction of N-Haloamide. VII. A Cleavage Reaction of Ether with N, N-Dihalobenzenesulfonamide. (2). Reactions of Tetrahydrofuran with N, N-Dibromobenzenesulfonamide, N-Bromosuccinimide, or Bromine. (1)
• Chemical Studies on Antibiotics produced by Actinomycetes. X. Racemomycin (7). Structure of Racemomycin-O
• Chemical Studies on Antibiotics produced by Actinomycetes. IX. Racemomycin. (6). Structure of New Degradation Product of Recemomycin-O
• Racemomycin (5). Degradation Products of Racemomycin-O.

もっと見る 閉じる

スポンサーリンク