Studies on Peptides. XXXII. The Use of N-Ethoxycarbonyl-2-ethoxy-1,2-dihydro-quinoline as a Coupling Reagent of Peptide-Fragments on Polymer Support
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概要
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As an example of peptide-fragment condensation on the polymer support, coupling reaction between Z (OMe)-Val-Lys (Z)-Val-Tyr-Pro-OH (positions 19 to 24 of ACTH) and H-Asp (OBzl)-Gly-resin and H-Ala-Gly-resin was performed. Among various coupling reagents so far examined, N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline gave relatively good results.
- 公益社団法人日本薬学会の論文
- 1971-09-25
著者
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河谷 紘樹
Faculty of Pharmaceutical Sciences, Kyoto University
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矢島 治明
Faculty Of Pharmaceutical Sciences Kyoto University
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