Reaction of Methyl 4,5-Epoxy-(2E)-pentenoate with Arenes. I. A Facile Synthesis of 4-Aryl-5-hydroxy-(2E)-pentenoate Derivatives
スポンサーリンク
概要
- 論文の詳細を見る
The reactivity of methyl 4,5-epoxy-(2E)-pentenoate (2) toward various aromatic nucleophiles in the presence of boron trifluoride etherate was examined. When benzene derivatives possessing an electron-donating substituent were employed, meta-substituted benzenes attacked only the 4-position of 2,while ortho- or para-substituted benzenes simultaneously attacked the 4- and 2-positions of 2.
- 社団法人日本薬学会の論文
- 1994-08-15
著者
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尾能 満智子
東邦大薬
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尾能 満智子
School Of Pharmaceutical Sciences Toho University
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山本 靖夫
School of Pharmaceutical Sciences, Toho University
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秋田 弘幸
School of Pharmaceutical Sciences, Toho University
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等々力 玲子
School of Pharmaceutical Sciences, Toho University
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山城 祐子
Faculty Of Pharmaceutical Sciences Kobe Gakuin University
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山本 譲
Faculty Of Pharmaceutical Sciences Kanazawa University
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Akita H
Toho Univ. Chiba Jpn
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秋田 弘幸
School Of Pharmaceutical Science Toho University
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Akita Hiroyuki
School Of Pharmaceutical Science Toho University
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Yamamoto Y
Tohoku Univ. Sendai Jpn
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Yamamoto Y
Pharmaceutical Research Laboratory Hokuriku Seiyaku Co. Ltd.
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Yamamoto Y
School Of Pharmaceutical Sciences Toho University
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等々力 玲子
School Of Pharmaceutical Sciences Toho University
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Yamamoto Yoshio
Pharmaceutical Research Division Takeda Chemical Industries Ltd.
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Yamamoto Y
大阪薬科大学
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Todoriki R
Toho Univ. Chiba Jpn
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山本 靖夫
School Of Pharmaceutical Sciences Toho University
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