Synthesis of Ozonolysis Products of Myxothiazol
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概要
- 論文の詳細を見る
By applying the Hantzsch thiazole procedure, the synthesis of bithiazole derivatives (2 and (±)-3) corresponding to degradation products of myxothiazol was achieved. Optically active (S)-3 (87-88% ee) and its analog (S)-16(91% ee) were obtained through enantioselective hydrolysis of the corresponding acetates ((±)-18,(±)-20 and (±)-21) using lipase in water-saturated organic solvent.
- 社団法人日本薬学会の論文
- 1994-06-15
著者
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秋田 弘幸
School of Pharmaceutical Sciences, Toho University
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南雲 紳史
School Of Pharmaceutical Science Toho University
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Nagumo S
School Of Pharmaceutical Science Toho University
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野澤 雅子
School of Pharmaceutical Science, Toho University
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Akita H
Toho Univ. Chiba Jpn
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秋田 弘幸
School Of Pharmaceutical Science Toho University
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Akita Hiroyuki
School Of Pharmaceutical Science Toho University
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Nozawa M
Graduate School Of Pharmaceutical Sciences Chiba University
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野澤 雅子
School Of Pharmaceutical Science Toho University
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Nagumo S
Hokkaido Coll. Pharmacy Otaru Jpn
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