A NEW SYNTHESIS OF EUPOLAURAMINE FROM A BENZ [f] INDOLE DERIVATIVE
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概要
- 論文の詳細を見る
Eupolauramine (1__-), a structurally unique alkaloid having oxindole and pyridine nuclei, was synthesized from a benz [f] indole derivative easily prepared from a pyrrole derivative. The synthetic route involves one-pot cnstruction of a pyridine ring via an enediamine moiety derived from the corresponding indole-2-carboxylic acid, and transformation of the enediamine to oxindole.
- 社団法人日本薬学会の論文
- 1988-09-25
著者
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渡辺 敏子
School Of Pharmaceutical Sciences Toho University
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横山 祐作
School of Pharmaceutical Sciences, Toho University
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村上 泰興
School of Pharmaceutical Sciences, Toho University
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Murakami Yukihisa
富山大学和漢医薬学総合研究所 複合薬物薬理学
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Murakami Yukihisa
Research Institute For Wakan-yaku (traditional Sino-japanese Medicines)
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酒井 正博
School Of Pharmaceutical Sciences Toho University
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Watanabe Toshifumi
Pharmaceutical Research Laboratories Ii Pharmaceutical Research Division Takeda Chemical Industries
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Watanabe T
Chiba Univ. Chiba Jpn
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Watanabe Toshihiro
Institute For Drug Discovery Research Yamanouchi Pharmaceutical Co. Ltd.
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村上 泰興
School Of Pharmaceutical Science Toho University
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