Synthetic Studies on Indoles and Related Compounds. XXV. The Friedel-Crafts Acylation of Ethyl 1H-Indole-2-carboxylate. (2)
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概要
- 論文の詳細を見る
The Friedel-Crafts acylation of ethyl 1H-indole-2-carboxylate (1) with various acylating reagents having a functional group or hetero atom and the acylation of some derivatives (6,7,8,and 9) of ethyl 1H-indole-2-carboxylate (1) with simple acylating reagents are described. Acylation occurred at the C_3-position or on the benzene moiety (mainly at the C_5-position) of the indole nucleus. The regioselectivity of the above acylation of indoles (1,6,7,8,and 9) is discussed.
- 社団法人日本薬学会の論文
- 1990-12-25
著者
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青木 剛
Fukushima Research Laboratories Toa Eiyo Ltd.
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福島 かおる
School Of Pharmaceutical Sciences Toho University
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谷 正宣
School of Pharmaceutical Sciences, Toho University
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青木 剛
School of Pharmaceutical Sciences, Toho University
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伊藤 貞雄
School of Pharmaceutical Sciences, Toho University
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松本 茂信
School of Pharmaceutical Sciences, Toho University
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秀嶋 麻美
School of Pharmaceutical Sciences, Toho University
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野澤 亮一
School of Pharmaceutical Sciences, Toho University
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前田 宜子
School of Pharmaceutical Sciences, Toho University
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田代 真由美
School of Pharmaceutical Sciences, Toho University
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横山 祐作
School of Pharmaceutical Sciences, Toho University
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村上 泰興
School of Pharmaceutical Sciences, Toho University
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野澤 亮一
School Of Pharmaceutical Sciences Toho University
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谷 正宣
School Of Pharmaceutical Sciences Toho University
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前田 宜子
School Of Pharmaceutical Sciences Toho University
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村上 泰興
東邦大・薬
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村上 泰興
School Of Pharmaceutical Science Toho University
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伊藤 貞雄
School Of Pharmaceutical Sciences Toho University
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秀嶋 麻美
School Of Pharmaceutical Sciences Toho University
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田代 真由美
School Of Pharmaceutical Sciences Toho University
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松本 茂信
School Of Pharmaceutical Sciences Toho University
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