Studies on Diazepines. VII. Syntheses of Novel 1H-1,2-Diazepines condensed with Aromatic Heterocyclic Rings

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概要

• 論文の詳細を見る

• Irradiation of the fused pyridinium ylides (6) or their dimers (7), prepared from 1,5-and 1,8-naphthyridine, thieno [2,3-b]- and thieno [3,2-b]-pyridine, and furo [2,3-b]-pyridine by N-amination with O-mesitylenesulfonylhydroxylamine followed by treatment with base, resulted in the fromation of the corresponding fused 1H-1,2-diazepines (8), which are previously unknown bicyclic ring systems. However, a similar synthetic route from the pyrrolopyridines (10) failed to yield pyrrolodiazepines.

• 社団法人日本薬学会の論文
• 1979-09-25

著者

• 沢西 啓之

  Faculty Of Pharmaceutical Sciences Hokuriku University

• 沢西 啓之

  School of Pharmacy, Hokuriku University

• 土屋 隆

  School of Pharmacy, Hokuriku University

• 円角 美智子

  School of Pharmacy, Hokuriku University

• 栗田 城治

  School of Pharmacy, Hokuriku University

• 栗田 城治

  Faculty of Pharmaceutical Sciences, Hokuriku University

• 土屋 隆

  Faculty Of Pharmaceutical Sciences Hokuriku University

• 栗田 城治

  Faculty Of Pharmaceutical Sciences Hokuriku University

• 円角 美智子

  School Of Pharmacy Hokuriku University

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