Reaction of Epoxides. V. 1,3-Dipolar Cycloaddition Reaction of Epoxides with Carbon-Nitrogen Double Bond Compounds

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概要

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• The reaction of epoxides with several conjugated C-N double bond compounds was attempted. Aromatic aldazines were found to undergo criss-cross cycloaddition toward epoxides. On the other hand, aromatic ketazines gave the oxazolidines formed by the cycloaddition of one molecule of epoxides to one of the C-N double bond of the ketazines. Moreover, in the reaction with N, N'-bis-benzylidene-p-phenylenediamine and N, N'-p-phenylene-bis-methylidenaniline, cycloaddition of two molecules of epoxides to two C-N double bonds of these compounds occurred to give the corresponding p-phenylenebis-oxazolidines.

• 公益社団法人日本薬学会の論文
• 1974-07-25

著者

• 古川 潮

  Faculty Of Pharmaceutical Sciences Kumamoto University

• 林 清五郎

  Faculty Of Pharmaceutical Sciences Kumamoto University

• 小島 洋子

  Faculty Of Pharmaceutical Sciences Kumamoto University

• 杉田 亮

  Faculty of Pharmaceutical Sciences, Kumamoto University

• 杉田 亮

  Faculty Of Pharmaceutical Sciences Kumamoto University

• 林清 五郎

  Faculty Of Pharmaceutical Sciences Kumamoto University

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