Arylthiation of Cyclohexanone Morpholine Enamine with Aryl Benzenethiosulfonates
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概要
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Sulfenylation of the nucleophilic β-carbon atom of 1-morpholino-1-cyclohexene with several thiosulfonates was attempted. Among these thiosulfonates, the reaction with alkyl alkanethiosulfonates and aralkyl benzenethiosulfonates were unsuccessful, but aryl benzenethiosulfonates in which an electron withdrawing group was substituted in the ortho or para position of the aryl group successfully reacted with 1-morpholino-1-cyclohexene to give the corresponding arylthio derivatives.
- 公益社団法人日本薬学会の論文
- 1973-09-25
著者
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古川 潮
Faculty Of Pharmaceutical Sciences Kumamoto University
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林 清五郎
Faculty Of Pharmaceutical Sciences Kumamoto University
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小島 洋子
Faculty Of Pharmaceutical Sciences Kumamoto University
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築地 制
Faculty of Pharmaceutical Sciences, Kumamoto University
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林清 五郎
Faculty Of Pharmaceutical Sciences Kumamoto University
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築地 制
Faculty Of Pharmaceutical Sciences Kumamoto University
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