Synthesis of Nucleosides and Related Compounds. XXXIV. Synthesis of 5-Isonitroso-1,3-dioxane-4,6-diones and Their Reactions

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概要

• 論文の詳細を見る

• Synthesis of 5-isonitroso-1,3-dioxane-4,6-dione (2 : isonitroso Meldrum's acid) and related compounds and their reactions were described. Compound (2) reacted with various alcohols to give hydroxyiminoacetic acid esters in moderate yields. Compound 2 was acetylated in the usual manner to give 5-acetoxyimino-1,3-dioxane-4,6-dione (9)as a stable crystalline substance, which acted not as a heterodiene but as a heterodienophile and underwent hetero Diels-Alder reaction with various dienes to form [4+2] adducts.

• 公益社団法人日本薬学会の論文
• 1994-06-15

著者

• 金子 主税

  東北大学

• 金子 主税

  Pharmaceutical Institute Medical Faculty University Of Tokyo

• 片桐 信弥

  Pharmaceutical Institute, Tohoku University

• 佐藤 弘

  Pharmaceutical Institute Tohoku University

• 片桐 信弥

  Health Sci. Univ. Hokkaido Hokkaido Jpn

• 片桐 信弥

  Pharmaceutical Institute Tohoku University

• 野地 弘之利

  Pharmaceutical Institute, Tohoku University

• 栗本 歩

  Pharmaceutical Institute, Tohoku University

• Katagiri N

  Pharmaceutical Institute Tohoku University

• 栗本 歩

  Pharmaceutical Institute Tohoku University

• 野地 弘之利

  Pharmaceutical Institute Tohoku University

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