抗HIV剤の創製を目標とした高度に修飾されたヌクレオシドの合成研究

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概要

• 論文の詳細を見る

• Recent studies on the synthesis of highly modified nucleosides, especially carbocyclic nucleosides, aiming at creating anti-HIV agents have been reviewed. The review includes new methods for the synthesis of carbocyclic C-nucleosides and carbocyclic N-nucleosides including carbocyclic oxetanocin and its analogues developed in our laboratory. Among the carbocyclic nucleosides synthesized, 9-(c-4,t-5-bishydroxymethylcyclopent-2-en-r-1-yl)-9H-adenine (BCA) showed significant anti-HIV activity.

• 公益社団法人日本薬学会の論文
• 1993-04-25

著者

• 片桐 信弥

  Health Sci. Univ. Hokkaido Hokkaido Jpn

• 片桐 信弥

  Pharmaceutical Institute Tohoku University

• 片桐 信弥

  東北大学薬学部

• Katagiri N

  Pharmaceutical Institute Tohoku University

関連論文

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