Reissert-Type Reaction of N-Sulfonyl- or N-Acyl-phthalazinimum Salts with Trimethyl Phosphite and Crystal Structure of Dimethyl 2-Mesyl-1,2-dihydro-1-phthalazinylphosphonate

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概要

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• Dimethyl 2-sulfonyl- and 2-acyl-1,2-dihydro-1-phthalazinylphosphonates (1a-e) were synthesized by the reaction of phthalazine with sulfonyl chloride or acyl chloride and trimethyl phosphite. The crystal structure of 1a was determined by X-ray analysis.

• 社団法人日本薬学会の論文
• 1990-06-25

著者

• 黒野 幸久

  神戸大学 大学院医学系研究科精神神経科学分野

• 八代 有

  Faculty of Pharmaceutical Sciences Nagoya City University

• 八代 有

  名古屋市立大学薬学部

• 黒野 幸久

  Faculty of Pharmaceutical Sciences, Nagoya City University

• 畑野 研一郎

  Faculty of Pharmaceutical Sciences, Nagoya City University

• 濱田 喜樹

  Faculty of Pharmacy, Meijo University

• 畑野 研一郎

  Faculty Of Pharmaceutical Sciences Nagoya City University

• 竹内 烈

  Faculty of Pharmacy, Meijo University

• 濱田 喜樹

  名城大学薬学部

• 竹内 烈

  名城大学薬学部

• 八代 有

  名古屋市立大学

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