Adsorption of Amino-acetamide Derivatives from 1-Octanol Solution by Silica Gel
スポンサーリンク
概要
- 論文の詳細を見る
Adsorption of amino-acetamide derivatives by silica gel from 1-octanol solution, the 1-octanol/water partition coefficient and the capacity factor were investigated. The physico-chemical parameters obtained were well correlated with each other. On the other hand, there was no correlation between the Hammett constant and adsorption parameters. The results indicate that adsorbability measurement may provide useful information for quantitative structure-activity relationship (QSAR) studies.
- 公益社団法人日本薬学会の論文
- 1984-10-25
著者
-
砂田 久一
Faculty Of Pharmacy Meijo University
-
杉浦 道治
Faculty of Pharmacy, Meijo University
-
濱田 喜樹
Faculty of Pharmacy, Meijo University
-
古川 圭子
Faculty Of Pharmacy Meijo University Yagoto-urayama
-
大塚 昭信
Faculty of Pharmacy, Meijo University
-
石野 隆三
Pharmaceutics Research Laboratory, Tanabe Seiyaku Co., Ltd.,
-
濱田 喜樹
名城大学薬学部
-
石野 隆三
Faculty of Pharmacy, Meijo University, Yagoto-Urayama
-
大塚 昭信
Faculty Of Pharmacy Meijo University
-
杉浦 道治
Faculty Of Pharmacy Meijo University
-
石野 隆三
Pharmaceutics Research Laboratory Tanabe Seiyaku Co. Ltd.
関連論文
- Regiospecific Nitration of Quinoline and isoquinoline through the Reissert Compounds
- Reissert-Type Reaction of N-Sulfonyl- or N-Acyl-phthalazinimum Salts with Trimethyl Phosphite and Crystal Structure of Dimethyl 2-Mesyl-1,2-dihydro-1-phthalazinylphosphonate
- Effect of Granule Strength on Compressed Tablet Strength
- Effect of Binder Characteristics on the Strength of Agglomerates Prepared by the Wet Method II
- Effect of Binder Characteristics on the Strength of Agglomerates Prepared by the Wet Method
- Computer Simulation of Agglomeration by a Two-Dimensional Random Addition Model. IV. : Agglomeration Kinetics and Micromeritic Properties of Agglomerate of Binary Mixtures of Adhesive Circles
- Reaction of Isoquinoline 2-Oxides with Methylsulfinylmethyl Carbanion
- Flocculation Kinetics of the Monodisperse System. II. Computer Simulation of Flocculation with Compaction by the Two-Dimensional Geometrical Random Coalescence Model
- Fundamental Study on the Evaluatoin of Strength of Granular Particles
- Influence of Moisture Adsorption of Volume Shrinkage and Diametral Tensile Strength of Sucrose Tablets
- Release of Sodium Guaiazurene-3-sulfonate from Polymer Film Dosage Forms
- Effect of Several Cellulosic Binders on Particle Size Distribution in Fluidized Bed Granulation
- Effect of Several Cellulosic Binders on Particle Size Distribution of Granules Prepared by a High-Speed Mixer
- Synthesis and Antimicrobial Activity of Salicylanilide Derivatives. II
- Influence of Compression Force on Consolidation Behavior and Drug Release Property of Wax Matrix Tablets
- Influence of Internal Structure on Kinetics of Drug Release from Wax Matrix Tablets
- Influence of Tabletting Speed on Compactibility and Compressibility of Two Direct Compressible Powders under High Speed Compression
- Release of Isosorbide Dinitrate from Polymer Film Dosage Forms and Absorption of This Drug through the Oral Mucosa of Rats
- Dissolution of Solid Dosage Form. VI. Dissolution of Nondisintegrating Single Component Tablets under Non-Sink Condition
- Hydrolysis of Acetylsalicylsalicylic Acid and Salicylsalicylic Acid in Aqueous Solution
- 14 Salicylanilide誘導体の除草作用について
- Salicylanilide誘導体の合成とその抗菌性について
- 2-Chloro-4-amino-5-(p-halogenophenoxy)phenylthiocyanate類の合成およびその抗菌性について(第1報)
- Influence of Fatty Acid-Alcohol Esters on Percutaneous Absorption of Hydrocortisone Butyrate Propionate
- Interactions between Water and Pharmaceutical Polymers Determined by Water-Vapor Sorption Measurement and Differential Scanning Calorimetry
- Release of Lidocaine from Polymer Film Dosage Forms
- Measurement of Adhesive Force between Particles of Organic Substances and Polymer Substrates by the Centrifugal Separation Method : Effect of Electrostatic Charge
- Solid-State Interaction of Ibuprofen with Polyvinylpyrrolidone
- Influence of the Molecular Weight of Binding Agents on the Physical Properties of Granules and Tablets
- Dissolution of Solid Dosage Form. IV. Equation for the Non-sink Dissolution of a Monodisperse System
- Measurement of the Adhesive Force between Particles and a Substrate by Means of the Impact Separation Method. Effect of the Surface Roughness and Type of Material of the Substrate
- Effect of Temperature on the Sticking of Low Melting Point Materials
- Pharmaceutical Preparations of Crude Drug Powder. III.The Effects of the Physical Properties of the Binder Solution on the Characteristics of the Granule from the Mixed Powders
- Absorption of Diltiazem in Beagle Dog from Pulsatile Release Tablet
- Design and Preparation of Pulsatile Release Tablet as a New Oral Drug Delivery System
- Adsorption of Amino-acetamide Derivatives from 1-Octanol Solution by Silica Gel
- Influence of Formulation Change on Drug Release Kinetics from Hydroxypropylmethylcellulose Matrix Tablets
- Studies on Application of Wax Matrix System for Controlled Drug Release
- Influence of Drug Solubility and Matrix Structure on Release Rate of Drugs from Wax Matrix Tablets
- Flocculation Kinetics of the Monodisperse System. Computer Simulation of Flocculation by the Two-Dimensional Geometrical Random Coalescence Model
- Dissolution of Solid Dosage Form. V. New Form Equations for the Non-sink Dissolution of a Monodisperse System
- Dissolution and Simulation Curved for Log-Normal Particle-Size-Distributed Model Systems
- Changes of Surface Area in the Dissolution Process of Crystalline Substances. V. : Dissolution and Simulation Curves for Log-Normal Particle-Size-Distributed Model Systems
- Changes of Surface Area in the Dissolution Process of Crystalline Substances. IV. Dissolution and Simulation Curves Estimated from Changes of Surface Area and Cube Root Law
- Changes of Surface Area in the Dissolution Process of Crystalline Substances. III. : Dissolution and Simulation Curves for Symmetrical Particle-Size-Distributed Model Systems
- Changes of Surface Area in the Dissolution Process of Crystalline Substances. II. : Dissolution and Simulation Curves for Mixed Systems of Sieved Particles
- 化学療法剤の研究(第5報) : アゾおよびジフェニールエーテル類などの線殺虫作用について
- ω-Aminosubstituted-acetanilide誘導体の合成とそれらの薬理作用
- Influence of Granulating Fluid Properties on Physical Properties of Kneading Mass and Granules
- Syntheses of Nitrogen-containing Heterocyclic Compounds. XLI. Reaction of Diazaphenanthrenes and Their N-Oxides with Methylsulfinyl Carbanion
- 含窒素複素環化合物の合成研究(第37報)2-Phenylquinoline 1-Oxide類およびPhenyl-1,8-naphthyridine類の合成とその抗菌性について
- 含窒素複素環化合物の合成研究(第32報)Nalidixic Acid類似のTriazaphenanthrene類の合成とDiazaphenanthrene類の抗菌性について
- キノリン誘導体について : その13 キノリン誘導体, アゾ化合物, ジフェニールエーテル類の抗いもち病作用について
- 含窒素複素環化合物の合成研究(第24報)5-Thiocyanato-6-haloquinaldine誘導体について
- Flocculation Studies of Granulated Stearyl Alcohol on the Surface of Aqueous Media. III. : Changes of Agglomerate Structure in a Two-Dimensional System with Anionic Surface-Acitive Agent
- Flocculation Kinetics of the Didisperse System-Computer Simulation of Flocculation by the Random Coalescence Model
- Carbanilide誘導体の合成とその抗菌性について
- 含窒素複素環化合物の研究-51-Phenanthroline N-OxideのReissert-Henze反応及びMeisenheimer反応について
- Preparation and Spectral Properties of 2-(2,4-Dichlorophenyl)-2-(1,2,3,5-tetrazol-1-ylmethyl)-1,3-dioxolan-4-ylmethanol and Its Benzoate and Methanesulfonate
- 含窒素複素環化合物の研究(第27報)3-Bromo Methylquinoline類の合成法
- Measurement of Adhesive Force between Particles and Polymer Films
- Effect of Particle Shape on the Compaction and Flow Properties of Powders
- Measurement of the Adhesive Force between Particles of Powdered Materials and a Glass Substrate by Means of the Impact Separation Method. III. : Effect of Particle Shape and Surface Asperity
- Measurements of the Adhesive Force between Particles of Powdered Organic Substances and a Glass Substrate by Means of the Impact Separation Method. II. Effect of Addition of Light Anhydrous Silicic Acid on the Adhesive Force of Potato Starch
- Dissolution of Solid Dosage Form. III. Equations for the Dissolution of a Nondisintegrating Single Component Tablet under a Nonsink Condition
- Dissolution of Solid Dosage Form. II. Equations for the Dissolution of Nondisintegrating Tablet under the Sink Condition
- ω-Aminosubstituted-acetamide誘導体の合成とその薬理作用
- ω-Aminosubstituted-acetamidodiphenyl Ether誘導体の合成とその薬用作用
- Evaluation of the Strength of a Scored Oblong Tablet
- cis-1-[2-Phenyl-4-(phenoxy or Phenylthio)methyl-1,3-dioxolan-2-ylmethyl]-1H-imidazole誘導体の合成とその抗菌作用について
- Influence of Granulating Fluids in Hydroxypropycellulose Binder Solution on Physical Properties of Lactose Granules
- Flocculation Studies of Granulated Stearyl Alcohol on the Surface of Aqueous Media. II. : Flocculation-Deflocculation Mechanism in a Two-Dimensional System
- Changes of Surface Area in the Dissolution Process of Crystalline Substances
- Synthesis of Naphtonaphthyridines by Skraup Reaction Using 3-Aminobenzo[g or h]quinoline
- 含窒素複素環化合物の研究(第47報)QuinolineからSpiro[cyclopropane-cyclopropa[c]quinoline]誘導体の生成について
- 含窒素複素環化合物の研究(第46報)Quinoline誘導体から1H-Benz[b]azepine誘導体への環転換について
- 含窒素複素環化合物の研究(第45報)Isoquinoline類を原料とするCyclopropa[c]isoquinoline誘導体の合成法
- 含窒素複素環化合物の研究(第43報)Pyridine誘導体を原料とし4級塩を経由するDicyclopropa[b, d](または[b, e])pyridine誘導体の2Step合成法
- Studies on Nitrogen-containing Heterocyclic Compounds. XL. Syntheses of 2-Alkylcyclopropa [c] quinolines
- 含窒素複素環化合物の研究(第35報)4-Amino-2-cyano-1,3-dimethoxy-1,2,3,4-tetrahydroisoquinoline類の合成とそれらの還元反応について
- 含窒素複素環化合物の研究(第39報)Quinoline誘導体を原料とし4級塩を経由するCyclopropa[c]quinoline誘導体の2Step合成法
- 含窒素複素環化合物の研究(第33報) Isoquinoline, 1,6-Naphthyridineを原料とする3-Alkoxyisoquinoline類, 7-, 8-置換-1,6-naphthyridineの合成法
- Moisture Sorption and Volume Expansion of Amorphous Lactose Tablets
- Syntheses of Nitrogen-containing Heterocyclic Compounds. XV. The Reissert Reaction of 1,6-Naphthyridine
- Measurements of the Adhesive Force between Particles of Powdered Organic Substances and a Glass Substrate by Means of the Impact Separation Method. I. Effect of Temperature
- Syntheses of Nitrogen-containing Heterocyclic Compounds. XXV. Chemical Reactivity of 4,6-Phenanthroline. (1)
- Quinoline誘導体を原料とするCyclopropa[c]quinoline誘導体の1Step合成法
- 含窒素複素環化合物の研究(第38報)Quinoline誘導体を原料としvon Braun反応を経由するCyclopropa[c]quinoline誘導体の2Step合成法
- 含窒素複素環化合物の研究(第36報)含窒素複素環化合物に対するvon Braun反応の改良とQuinaldineからの3-Bromoquinaldineの合成法
- Studies on Nitrogen-containing Heterocyclic Compounds. XXXIV. Chemical Reactivity of 1 (or 2)-Cyano-1,2-dihydro (iso)-quinolines and 1 (or 2)-Cyano-1,2,3,4-tetrahydro (iso) quinolines
- 含窒素複素環化合物の研究(第31報)2-Bromobenzo[f]quinolineおよびその関連化合物の合成と化学反応性
- Syntheses of Nitrogen-containing Heterocyclic Compounds. XXIII. Reaction of Naphthyridine Derivatives, with Special Reference to that of 1,7-Naphthyridine
- Synthesis of Nitrogen-containing Heterocyclic Compounds. XX. Improvement of One-step Synthesis of Phenanthrolines and Some Reactions of 4,6-Phenanthroline
- Syntheses of Nitrogen-containing Compounds. XVIII. Syntheses of Naphthyridines by Improved One-Step Process
- Syntheses of Nitrogen-containing Compounds. XVII. Improvement of One-Step Synthesis of Naphthyridine Derivatives and Their Methylation with Dimethyl Sulfoxide in the Presence of Base
- Sustained Release Mechanisms of Wax Matrix System for Controlled Release
- Computer Simulation of Agglomeration by a Two-dimensional Random Addition Model. III. -Agglomeration Kinetics and Micromeritic Properties of Closely-packed Agglomerates of Heterogeneous Binary Circles-
- Simulation of Agglomeration. II. Two-dimensional Random Addition Model. (1)
- Caking of δ-D-Gluconolactone Powder
- Studies on Compaction of Powders. III. Compression Behavior of Several Powders under Low Pressure