A Simple Synthesis of 1,3-Dialkylpyrido [2,3-d] pyrimidines
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概要
- 論文の詳細を見る
A new and convenient synthesis of 1,3-dialkylpyrido [2,3-d] pyrimidine-2,4 (1H, 3H)-diones from 6-allylamino-and 6-(substituted allyl) aminouracils by PdCl_2-CuCl-O_2-catalyzed oxidative cyclization is described. Further, 1,3-dimethylpyrido [2,3-d] pyrimidine 2,4 (1H, 3H)-dione (4a) was prepared by the reaction of 6-allylamino-1,3-dimethyluracils (3a) with (AcO)_2 Pd and by the thermal cyclization of 3a.
- 社団法人日本薬学会の論文
- 1985-04-25
著者
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小倉 治夫
School of Pharmaceutical Sciences, Kitasato University
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小倉 治夫
School Of Pharmaceutical Sciences Kitasato University
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川原 徳夫
Hokkaido Institute of Pharmaceutical Sciences
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渡辺 恭一
Sloan-kettering Instiute For Cancer Research Memorial Sloan-kettering Cancer Center:sloan-kettering
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伊東 常男
School Of Pharmaceutical Sciences Kitasato University
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中嶋 孝子
Hokkaido Institute of Pharmaceutical Sciences
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WATANABE KYOICHI
Sloan-Kettering Institute for Cancer Research, Sloan-Kettering Division of Graduate School of Medica
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川原 徳夫
北海道薬大
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Watanabe Kyoichi
Sloan-kettering Institute For Cancer Research Memorial Sloan-kettering Cancer Center Sloan-ketting D
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