Synthesis of Polycyclines. II. Synthesis of 12-Hydroxy-5a, 6,-7,8,9,10,11,11a-octahydro-5 (12H)-naphthacenones

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概要

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• A convenient synthesis is reported of 1-substituted 7,8,9,10-tetrahydro-5,12-naphthacenediones (3a-d) and 4-substituted 12-hydroxy-5a, 6,7,8,9,10,11,11a-octahydro-5 (12H)-naphthacenones (4a-c) by means of the Diels-Alder reaction of 1,4-naphthoquinones (1a-d) with 1,2-dimethylenecyclohexane, followed by aromatization through dehydrogenation (3a-d) or by catalytic hydrogenation (4a-c).

• 公益社団法人日本薬学会の論文
• 1979-09-25

著者

• 織田 範一

  Faculty of Pharmaceutical Sciences, Nagoya City University

• 伊藤 磯雄

  Faculty of Pharmaceutical Sciences, Nagoya City University

• 永井 慎一

  Faculty of Pharmaceutical Sciences, Nagoya City University

• 伊藤 磯雄

  名古屋市立大学薬学部

• 織田 範一

  Faculty Of Pharmaceutical Sciences Nagoya City University

• 伊藤 磯雄

  Faculty Of Pharmaceutical Sciences Nagoya City University

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