Transformation of Pyrazolo [3,4-c] [1,5] benzothiazepines into Quinolines
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概要
- 論文の詳細を見る
Pyrazolo [3,4-c] [1,5] benzothiazepines (4,5) were transformed into quinolines (6,7) in refluxing xylene in the presence of sodium hydride. The reaction of 6 with N, N-dimethylformamide dimethylacetal gave 1-methyl-4-oxo-3-phenyl-1,2,3,4-tetrahydropyrimido [5,4-b]-quinoline (10). The photochemical reaction of 4-anilino-2,3-dimethyl-1-phenyl-3-pyrazolin-5-one (12) in xylene under a 100 W high pressure Hg-lamp gave 1,2-dihydro-1-methyl-3-oxo-2-phenyl-3H-pyrazolo [4,3-b] quinoline (3).
- 公益社団法人日本薬学会の論文
- 1984-04-25
著者
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織田 範一
Faculty of Pharmaceutical Sciences, Nagoya City University
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植田 泰誠
Faculty of Pharmaceutical Sciences, Nagoya City University
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永井 慎一
Faculty of Pharmaceutical Sciences, Nagoya City University
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榊原 仁作
名市大院薬
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榊原 仁作
Faculty Of Pharmaceutical Sciences Science University Of Tokyo
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永井 慎一
名市大薬
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織田 範一
Faculty Of Pharmaceutical Sciences Nagoya City University
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植田 泰誠
Faculty Of Pharmaceutical Sciences Nagoya City University
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榊原 仁作
Faculty Of Pharmaceutical Sciences Nagoya City University
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