The Reactions of Activated Amides. V. The Reactions of Cyclic Amide Acetals with Electrophiles

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概要

• 論文の詳細を見る

• The condensations of 1-methyl-2-piperidone diethylacetal (VI) and 1-methyl-2-pyrrolidone dimethylacetal (XX) with several electrophiles were carried out and it was found that VI afforded the 3,3-disubstituted compounds. When benzyl chloride was used, even the compound VI afforded the 3-monosubstituted compounds. The mechanism for this anomaly is discussed.

• 公益社団法人日本薬学会の論文
• 1972-08-25

著者

• 伴 義雄

  Faculty of Pharmaceutical Sciences, School of Medicine, Hokkaido University

• 大石 武

  Faculty Of Engineering Yokohama National University:(present Address)meiji College Of Pharmacy

• 森 美和子

  北大・薬

• 伴 義雄

  東邦大・薬

• 伴 義雄

  Faculty Of Pharmaceutical Sciences Hokkaido University

• 大石 武

  北大・薬:(現)理化学研究所

• 森 美和子

  Faculty of Pharmaceutical Sciences, Hokkaido University

• 中木村 宏

  Faculty of Pharmaceutical Sciences, Hokkaido University

• 中木村 宏

  Faculty Of Pharmaceutical Sciences Hokkaido University

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