Potential Antimetabolites. III. Synthesis of 5-Aminoimidazole-4-carboxthioamide and Nitro-1-β-D-ribofuranosylimidazoles.
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概要
- 論文の詳細を見る
5-Aminoimidazole-4-carboxthioamide was synthesized by the phosphorus pentasul-fide-pyridine treatment of 5-aminoimidazole-4-carboxamide. The structure was elucidated both by chemical and physical means. 1-β-D-Ribofuranosyl-4-methyl-5-nitro-imidazole and 1-β-D-ribofuranosyl-4-nitro-5-methoxycarbonylimidazole were synthesized by the condensation of appropriate imidazole chloro-mercury salt with 2,3,5-tri-O-benzoyl-D-ribofuranosyl chloride followed by the removal of protecting groups.
- 公益社団法人日本薬学会の論文
- 1962-08-25
著者
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池原 森男
Faculty of Pharmaceutical Sciences, Osaka University(Present address)
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中沢 信彦
Faculty Of Pharmaceutical Sciences School Of Medicine Hokkaido University.
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池原 森男
Faculty Of Pharmaceutical Sciences Osaka University
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中山 熙士
Faculty of Pharmaceutical Sciences, School of Medicine, Hokkaido University.
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中山 熙士
Faculty Of Pharmaceutical Sciences School Of Medicine Hokkaido University.
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