Studies on Pyrimidine Derivatives and Related Compounds. LXXXI. Reactions of Aryl Isothiocyanates with Thiamine and Related Thiazolium Ylides
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概要
- 論文の詳細を見る
Reactions of thiamine and related thiazolium ylides with aryl isothiocyanates afforded zwitterionic adducts (Va-j) or cycloadducts (VIa-c). An electron attracting substituent in the aryl group favored the zwitterion formation, while an electron donating substituent favored the cycloadduct formation. A ring expansion reaction of 2-thiocarbamoylated thiazolium ring giving 1,4-thiazine derivative was also described.
- 公益社団法人日本薬学会の論文
- 1974-02-25
著者
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高見沢 映
Shionogi Research Laboratory, Shionogi & Co., Ltd.
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高見沢 映
新潟薬科大学
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酒井 昇二
Shionogi Research Laboratory, Shionogi & Co., Ltd.
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高見沢 映
Shionogi Research Laboratory Shionogi & Co. Ltd.
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酒井 昇二
Shionogi Research Laboratory Shionogi And Co. Ltd.
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酒井 昇二
Shionogi Research Laboratory Shionogi & Co. Ltd.
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松本 佐市
Shionogi Research Laboratory, Shionogi and Co., Ltd.
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松本 佐市
Shionogi Research Laboratory Shionogi And Co. Ltd.
関連論文
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- Studies on Pyrimidine Derivatives and Related Compounds. XLVI. The Reactions of Diethyl Acetylphosphonate with Thiamine : Takamizawa Reaction (5).
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