Studies on the Pyrimidine Derivatives and Related Compounds. XL. Reaction of 3-Benzyl-4-methyl-5-(2-hydroxyethyl)thiazolium Salts with Diethyl Benzoylphosphonate

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概要

• 論文の詳細を見る

• Reaction of 3-benzyl-4-methyl-5-(2-hydroxyethyl)thiazolium chloride (V) with diethyl benzoylphosphonate (VII) was studied successively as an analogue of thiamine. It is also appeared in this case that a novel reaction took place accompanied by the ring expansion from thiazole to 1,4-thizzine ring.

• 社団法人日本薬学会の論文
• 1966-07-25

著者

• 佐藤 義朗

  Shionogi Research Laboratory Shionogi & Co. Ltd.

• 高見沢 映

  Shionogi Research Laboratory, Shionogi & Co., Ltd.

• 高見沢 映

  Niigata College Of Pharmacy

• 高見沢 映

  Shionogi Research Laboratory Shionogi & Co. Ltd.

関連論文

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• Studies on Pyrimidine Derivatives and Related Compounds. XLVII. Reaction of Thiamine with Dialkyl Acylphos-phonates or Methyl Phenylacyl-phosphinates : Takamizawa Reaction 6
• Studies on Pyrimidine Derivatives and Related Compounds. XLVI. The Reactions of Diethyl Acetylphosphonate with Thiamine : Takamizawa Reaction (5).
• Studies on the Pyrimidine Derivatives and Related Compounds. XL. Reaction of 3-Benzyl-4-methyl-5-(2-hydroxyethyl)thiazolium Salts with Diethyl Benzoylphosphonate
• 41.ピリミジン誘導体および関連化合物の研究(LVI) : ビタミンB_1とリン誘導体との反応(5)(第18回大会研究発表要旨)
• Studies on the Pyrimidine Derivatives and Related Compounds. XXXIX. On the Oxidation Products of 2-Pheny1-4-(2-methyl-4-amino-5-pyrimidyl)methyl-5-methyl-6-(2-benzoyloxy or hydroxy)-ethyl-4H-1,4-thiazin-3(2H)-one
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