Studies on the Pyrimidine Derivatives and Related Compounds. XXXV. On the Reaction Product of Thiamine with Diethyl Benzoylphosphonate
スポンサーリンク
概要
- 論文の詳細を見る
It was shown that a new thiamine derivative which was obtained from the reaction of the neutral form of thiamine (I) with diethyl benzoylphosphonate (II) should be formulated as 2-phenyl-3-oxo-4-(2-methyl-4-amino-5-pyrimidyl) methyl-5-methyl-6-(2-benzoyloxy) ethyl-2,3-dihydro-4H-1,4-thiazine (IV). A novel benzoylation reaction accompanied by the rearrangement from thiazole to 1,4-thiazine is also described.
- 社団法人日本薬学会の論文
- 1966-04-25
著者
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高見沢 映
Shionogi Research Laboratory, Shionogi & Co., Ltd.
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田中 幸子
Shionogi Research Laboratory, Shionogi & Co., Ltd.
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田中 幸子
塩野義研究所
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佐藤 義郎
Shionogi Research Laboratory, Shionogi & Co., Ltd.
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伊藤 寿子
Shionogi Research Laboratory, Shionogi & Co., Ltd.
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高見沢 映
Shionogi Research Laboratory Shionogi & Co. Ltd.
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佐藤 義郎
Shionogi Research Laboratory Shionogi & Co. Ltd.
関連論文
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- Studies on Pyrimidine Derivatives and Related Compounds. XLVII. Reaction of Thiamine with Dialkyl Acylphos-phonates or Methyl Phenylacyl-phosphinates : Takamizawa Reaction 6
- Studies on Pyrimidine Derivatives and Related Compounds. XLVI. The Reactions of Diethyl Acetylphosphonate with Thiamine : Takamizawa Reaction (5).
- Studies on the Pyrimidine Derivatives and Related Compounds. XL. Reaction of 3-Benzyl-4-methyl-5-(2-hydroxyethyl)thiazolium Salts with Diethyl Benzoylphosphonate
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- 7.Benzothiamine(VI)(第154回会議研究発表要旨)
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- 7.ビタミンB_1新誘導体について(第149回会議研究発表要旨)
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