Syntheses of Pyrazole Derivatives. XI. Acetylation Products of 7-Aminopyrazolo [1,5-a] pyrimidines. Supplement
スポンサーリンク
概要
- 論文の詳細を見る
In connection with the study of the acetylation of 7-aminopyrazolo [1,5-a] pyrimidines, further studies on the acetylation were investigated. Mono- and diacetates were obtained from the compounds being substituted with methyl-, Phenyl-, or ethoxy-carbonyl group at the C-6 position and only monoacetates being unsubstituted or with a cyano group at the C-6 position. The reason for this was confirmed to be the steric effect of the substituents at the C-6 position. Various 7-acylamino (XXXVII〜XL, XLII〜XLVI), 7-alkylamino (XLI, LVIII〜LXVI), and 7-H pyrazolo [1,5-a] pyrimidines (LIII〜LV) were also derived.
- 公益社団法人日本薬学会の論文
- 1965-10-25
著者
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浜島 好男
Shionogi Research Laboratory Shionogi & Co. Ltd.
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高見沢 映
Shionogi Research Laboratory Shionogi & Co. Ltd.
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