Studies on Steroid Conjugates. II. Synthesis of 16-Epiestriol Monoglucuronides
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概要
- 論文の詳細を見る
16-Epiestriol 16- and 17-monoglucuronides (XI, V) were prepared from 3-benzyloxy-17β-hydroxyestra-1,3,5 (10)-trien-16-one (I) employing Koenigs-Knorr reaction as shown in Chart 1. These synthetic glucuronides readily underwent hydrolysis with beef-liver β-glucuronidase preparation to furnish 16-epiestriol and free glucuronic acid.
- 公益社団法人日本薬学会の論文
- 1969-08-25
著者
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南原 利夫
Pharmaceutical Institute, Tohoku University
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松木 容彦
Pharmaceutical Institute, Tohoku University
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松木 容彦
Pharmaceutical Institute Tohoku University
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千葉 智巳
Pharmaceutical Institute, Tohoku University
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千葉 智巳
Pharmaceutical Institute Tohoku University
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南原 利夫
Pharmaceutical Institute Tohoku University
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