Synthesis in the Diazasteroid Group. XVIII. Syntheses of the 9,17-Diazasteroid System

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概要

• 論文の詳細を見る

• A 9,17-diazasteroid system, I, was synthesized from an aminoester, III, and cyclohexanone. Unfortunately the yield was poor. Another 9,17-diazasteroid system, II, was prepared from the condensation product, XVa, of quinoline N-oxide with an active methine compound, IV. Thus, XVa was hydrolyzed, followed by decarboxylation, reduction and cyclization. The yield in each step to II was moderate.

• 公益社団法人日本薬学会の論文
• 1982-04-25

著者

• 高畑 廣紀

  富山医科薬科大学薬学部

• 平井 美朗

  Faculty of Pharmaceutical Sciences, Toyama Medical and Pharmaceutical University

• 高畑 広紀

  Faculty of Pharmaceutical Sciences, Toyama Medical & Pharmaceutical University

• 的場 勝英

  Faculty Of Pharmaceutical Sciences Toyama Medical & Pharmaceutical University

• 的場 勝英

  Faculty Of Pharmaceutical Sciences Osaka University

• 平井 美朗

  富山医科薬科大学薬学部

• 平井 美朗

  Pharmaceutical Institute Tohoku University

• 高畑 広紀

  Faculty Of Pharmaceutical Sciences University Of Tokyo

• 山崎 高応

  富山医科薬科大学 薬

• 山崎 高応

  Faculty of Pharmaceutical Sciences

• 福島 明子

  Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University

• 平井 美朗

  Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University

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