The Chemistry of Lactim Ethers. II. Reaction of Lactim Ethers with 2-Carbethoxymethyl Piperidines

スポンサーリンク

概要

• 論文の詳細を見る

• Annulation reactions of methyl valelolactim (2) and methyl caprolactim (3) with cyclic β-aminoesters, such as 2-carbethoxymethyl piperidine derivatives (4 or 5), often gave two kinds of products apparently arising from the imine and enamine forms of 2 and 3. These chemical properties were consistent with NMR observations of lactim ethers in CD_3OD solution.

• 公益社団法人日本薬学会の論文
• 1980-01-25

著者

• 山崎 高應

  Faculty of Pharmaceutical Sciences, University of Toyama

• 高畑 廣紀

  富山医科薬科大学薬学部

• 山崎 高應

  Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University

• 高畑 広紀

  Faculty of Pharmaceutical Sciences, Toyama Medical & Pharmaceutical University

• 石倉 稔

  Faculty Of Pharmaceutical Sciences Higashi-nippon-gakuen University

• 石倉 稔

  Faculty Of Pharmaceutical Sciences

• 高畑 広紀

  Faculty Of Pharmaceutical Sciences University Of Tokyo

関連論文

• Synthetic Studies of Azaflavonoids. I. Studies on the Synthesis of 5-Azaflavone
• 8,13-Diazagona-1,3,5 (10)-triene-12-ones, Synthesis and Stereochemistry
• A Stereocontrolled Synthesis of (±)-Emetine and (±)-Protoemetinol by Intramolecular Michael Reaction
• Chemistry of 2-Methoxy-2,5-cyclohexadienone. V. Photochemical Rearrangement and Oxidation of 2-Methoxy-4-methyl-4-phenyl-2-cyclohexenone and 2-Methoxy-4-methyl-4-phenyl-2,5-eyclohexadienone(Organic,Chemical)
• 薬理活性志向のヘテロ環の合成研究
• Synthesis in the Diazasteroid Group. XX. Synthesis of the 5,14-Diazasteroid System(Organic,Chemical)
• チオアミド官能基の特性を利用する複素環合成
• An Efficient Total Synthesis of (±)-Epilupinine and (±)-Lupinine from a Common Quinolizidine Intermediate
• Favorskii Reaction of 2-Bromobicyclo[3.3.1]nonan-3-one
• Reaction of Aliphatic Dicarboxylic Acids with Acyl Chlorides in the Presence of Aluminum Chloride
• Ketene-S, N-acetals as Synthetic Intermediates for Heterocycles. Reaction of Ketene-S, N-acetals with Aryl Isocyanates
• Chemistry of 2-Methoxy-2,5-cyclohexadienone. IV. Photochemistry of 2-Methoxy-4,4-diphenyl-2,5-cyclohexadienone and 4-Dichloromethyl-2-methoxy-4-methyl-2,5-cyclohexadienone
• Reduction of Vinylogous Thioesters with Lithium Aluminum Hydride. II. Reduction of 2-Methyl-3-phenylthio-5-substituted-2-cyclopentenones
• Reduction of Vinylogous Thioesters with Lithium Aluminum Hydride. I. Reduction of β-Phenylthio-α, β-unsaturated Cyclic Ketones
• Chemistry of 2-Methoxy-2,5-cyclohexadienones. III. Syntheses of 2-Methoxy-4,4-diphenyl-2,5-cyclohexadienone and 4-Dichloromethyl-2-methoxy-4-methyl-2,5-cyclohexadienone
• Structural Modification of Bioactive Compounds. II. Syntheses of Aminophosphonoic Acids
• Chemistry of 2-Methoxy-2,5-cyclohexadienones. II. Oxidation of 2-Methoxy-4,4-dimethyl-2,5-cyclohexadienone
• Synthesis in the Diazasteroid Group. XXI. An Alternative Synthesis of the 8,16-Diazasteroid System
• KETENE-S, N-ACETALS AS SYNTHETIC INTERMEDIATES FOR HETEROCYCLES. A NOVEL SYNTHESIS OF POLYFUNCTIONALIZED PYRIDINE-2-THIONES
• Structural Modification of Bioactive Compounds. I. Syntheses of Vitamin D Analogues I
• Nitration of 2-Cyclohexenone Derivatives and Some Reactions of the Products
• AN EASY SYNTHESIS OF MONOMETHYL MALONATE DERIVATIVES
• 63 Pd触媒による一酸化炭素挿入反応を利用した1,4-Benzodiazepine骨格の合成並びにその天然物合成への応用
• Activated Lactams. VI. The Cycloaddition Reaction of Cyclic Ketene-S, N-acetals with Dimethyl Acetylenedicarboxylate
• A Novel Synthesis of 4-Aryl-and 4-Heteroarylpyridines via Diethyl (4-pyridyl) borane
• New Synthesis of Pyrrolo-1,4-benzodiazepines by Utilizing Palladium-Catalyzed Carbonylation
• Dialkyl (3-pyridyl) boranes
• 36 Pd触媒による一酸化炭素挿入反応を用いた天然物の合成
• The Chemistry of Lactim Ethers. IV. Syntheses of 1,9-and 5,9-Diazasteroid Systems
• The Chemistry of Lactim Ethers. II. Reaction of Lactim Ethers with 2-Carbethoxymethyl Piperidines
• Acid-catalyzed Cyclization of Chalcones derived from Various Nitrogenous Heteroaromatic Compounds. II
• Chemistry of 2-Methoxy-2,5-cyclohexadienones. I. Photochemistry of 2-Methoxy-4,4-dimethyl-2,5-cyclohexadienone
• A FACILE SYNTHESIS OF 2-METHOXY-4,4-DIMETHYL-2,5-CYCLOHEXADIENONE VIA 5,5-DIMETHYL-2-NITRO-1,3-CYCLOHEXADIENOL
• Michael Addition of [1H] Pyrrole
• Synthesis in the Diazasteroid Group. XIX. Synthesis of the 9,13-Diazasteroid System
• The Chemistry of Lactim Ethers. V. Reaction of Lactim Thioethers with β-Aminoesters
• Acid-catalyzed Cyclization of Chalcones derived from Various Nitrogenous Heteroaromatic Compounds
• A Convenient Synthesis of Monocyclic β-Lactams by Means of Solid-Liquid Phase Transfer Reactions
• Synthesis in the Diazasteroid Group. XV. Syntheses of the 5,9- and 8,13-Diazasteroids
• Synthesis in the Diazasteroid Group. XIV. Synthesis of the 13,15-Diazasteroid System
• Reaction of Lactim Thioethers with 1-Carbethoxymethyl-1,2,3,4-tetrahydroisoquinoline
• Synthesis of 8,10-Diaza-estrane
• Synthetic Studies of Azaflavonoids. II. Synthesis of 6-Azaflavonoids
• Studies on O-Alkylated Imides. II. Some Reactions of O-Ethyl Succinimide and O-Ethyl 4,4-Dimethyl-glutarimide
• Reduction of O-Alkylated Imides
• Synthesis of Zwitterionic Pyridazine Derivatives. I
• Synthesis in the Diazasteroid Group. XVIII. Syntheses of the 9,17-Diazasteroid System
• Synthesis in the Diazasteroid Group. XVII. Syntheses of the 4,11-Diazasteroid System
• New Synthetic Routes to Carbohydrates by the Use of Telomers of Vinylene Carbonate with Polyhalomethanes
• チオアミド官能基の特性を利用する複素環合成
• 二重不斉化反応による光学純度累進効果を活用する有機合成
• 非キラルなクロマトグラフィーにおける光学分割現象
• 高選択的なヘテロ環化反応の開発と生物活性物質の合成への応用
• 2級アリルアルコールに対する分子内アミノ付加反応を基盤とする含窒素生物活性物質のキラル合成

もっと見る 閉じる

スポンサーリンク