Synthesis of Oxapenam Derivatives
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概要
- 論文の詳細を見る
Photolysis of N-diazoacetyloxazolidine compounds, 7c and 8c, afforded oxapenams, 9 and 10,respectively. The physical data of 9 and 10 along with their behavior on thinlayer chromatograms were consistent with that of the samples derived from clavulanic acid (1), a β-lactamase inhibitor, confirming their structures. Further, a methylene oxapenam 18 was obtained from an oxapenam 17 having a phenylseleno group by selenoxide elimination reaction.
- 社団法人日本薬学会の論文
- 1978-02-25
著者
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大木 英二
Central Research Laboratories, Sankyo Co., Ltd.
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老田 貞夫
Central Research Laboratories, Sankyo Co., Ltd.
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吉田 明
Central Research Laboratories, Sankyo Co., Ltd.
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吉田 明
Chemical Research Laboratories Sankyo Co. Ltd.
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老田 貞夫
Medicinal Chemistry Research Laboratories, Sankyo Co., Ltd.,
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大木 英二
Research Laboratory Zenyaku Kogyo Co. Ltd.
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大木 英二
Central Research Laboratories Sankyo Co. Ltd.
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老田 貞夫
Medicinal Chemistry Research Laboratories Sankyo Co. Ltd.
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