Enantiocontrolled Synthesis of the Antifungal β-Lactam (2R, 5S)-2-(Hydroxymethyl)clavam
スポンサーリンク
概要
- 論文の詳細を見る
The antifungal β-lactam (2R, 5S)-2-(hydroxymethyl)clavam was synthesized in a convergent and stereocontrolled manner from methyl 6-phthalimidopenicillanate and 2,3-O-isopropylidene-(R)-glyceraldehyde. Convenient methods of acetonide cleavage and phthalimide deblocking are also described.
- 公益社団法人日本薬学会の論文
- 1991-09-25
著者
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鴻巣 俊之
Medicinal Chemistry Research Laboratories, Sankyo Co., Ltd.,
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老田 貞夫
Medicinal Chemistry Research Laboratories, Sankyo Co., Ltd.,
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老田 貞夫
Medicinal Chemistry Research Laboratories Sankyo Co. Ltd.
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鴻巣 俊之
Medicinal Chemistry Research Laboratories Sankyo Co. Ltd.
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鴻巣 俊之
Medicinal Chemistry Res. Laboratories Ii Daiichi Sankyo Co. Ltd.
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