Triazole Antifungals. V. Synthesis and Antifungal Activities of Some Amides Related to 3-Acylamino-2-aryl-1-triazolyl-2-butanol

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概要

• 論文の詳細を見る

• Amides, 2 and 3,related to the potent antifungal triazole-amide 3-acylamino-2-aryl-1-triazolyl-2-butanol (1) were synthesized starting from the triazole-alcohol 6. The antifungal activity of 2 and 3 aganist a mouse systemic Candida albicans infection was found to be less potent than that of 1.

• 公益社団法人日本薬学会の論文
• 1992-03-25

著者

• 安田 紘

  Biological Research Laboratories Sankyo Co. Ltd.

• 田中 輝夫

  Medical Chemistry Research Laboratories Sankyo Co. Ltd.

• 鴻巣 俊之

  Medicinal Chemistry Research Laboratories, Sankyo Co., Ltd.,

• 老田 貞夫

  Medicinal Chemistry Research Laboratories, Sankyo Co., Ltd.,

• 武田 憲子

  Medicinal Chemistry Research Laboratories Sankyo Co., Ltd.

• 武田 憲子

  Medical Chemistry Research Laboratories Sankyo Co. Ltd.

• Konosu Toshiyuki

  Medicinal Chemistry Research Laboratories II, Daiichi Sankyo Co., Ltd.

• 老田 貞夫

  Medicinal Chemistry Research Laboratories Sankyo Co. Ltd.

• 鴻巣 俊之

  Medicinal Chemistry Research Laboratories Sankyo Co. Ltd.

• 鴻巣 俊之

  Medicinal Chemistry Res. Laboratories Ii Daiichi Sankyo Co. Ltd.

• Konosu Toshiyuki

  Medicinal Chemistry Res. Laboratories Ii Daiichi Sankyo Co. Ltd.

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