PAYNE REARRANGEMENT ROUTE TO THE OPTICALLY ACTIVE OXIRANE PRECURSOR FOR THE PREPARATION OF TRIAZOLE ANTIFUNGALS
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概要
- 論文の詳細を見る
Optically active epoxide 1,an important intermediate for the preparation of antifungal triazole-amides 2,was synthesized starting from the (S)-lactic acid- derived ketone 9 and taking advantage of the Payne rearrangement of the epoxyalocohol 8.
- 社団法人日本薬学会の論文
- 1992-02-25
著者
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宮岡 武男
Medicinal Chemistry Research Laboratories Sankyo Co. Ltd.
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鴻巣 俊之
Medicinal Chemistry Research Laboratories, Sankyo Co., Ltd.,
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田島 和
Medicinal Chemistry Research Laboratories, Sankyo Co., Ltd.,
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老田 貞夫
Medicinal Chemistry Research Laboratories, Sankyo Co., Ltd.,
-
田島 和
Medicinal Chemistry Research Laboratories Sankyo Co. Ltd.
-
老田 貞夫
Medicinal Chemistry Research Laboratories Sankyo Co. Ltd.
-
鴻巣 俊之
Medicinal Chemistry Research Laboratories Sankyo Co. Ltd.
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鴻巣 俊之
Medicinal Chemistry Res. Laboratories Ii Daiichi Sankyo Co. Ltd.
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