Synthesis of 5,8-Dihydroxy-3,4-dihydrocarbostyril

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概要

• 論文の詳細を見る

• 5,8-Dihydroxy-3,4-dihydrocarbostyril, a key intermediate for the synthesis of β_1-selective 8-acetonyloxy-5-[3-(3,4-dimethoxyphenethylamino)-2-hydroxypropoxy]-3,4-dihydrocarbostyril hydrochloride (opc-1427) was prepared from 2,5-dimethoxyaniline.

• 社団法人日本薬学会の論文
• 1981-08-25

著者

• 中川 量之

  2nd Tokushima Institute Of New Drugs Research Otsuka Pharmaceutical Co. Ltd.

• 中川 量之

  大塚製薬株式会社有機化学研究所

• 中川 量之

  大塚製薬株式会社徳島研究所

• 楊 永雄

  Tokushima Research Institute, Otsuka Pharmaceutical Co., Ltd.,

• 富永 道明

  Laboratories of Medicinal Chemistry

• 中川 量之

  Laboratories of Medicinal Chemistry

• 楊 永雄

  Laboratories of Medicinal Chemistry, Tokushima Research Institute, Otsuka Pharmaceutical Co., Ltd.

• 大崎 正明

  Laboratories of Medicinal Chemistry, Tokushima Research Institute, Otsuka Pharmaceutical Co., Ltd.

• 真鍋 義明

  Laboratories of Medicinal Chemistry, Tokushima Research Institute, Otsuka Pharmaceutical Co., Ltd.

• 真鍋 義明

  Laboratories Of Medicinal Chemistry Tokushima Research Institute Otsuka Pharmaceutical Co. Ltd.

• 富永 道明

  大塚製薬(株)徳島新薬第二研究所

• 楊 永雄

  Tokushima Research Institute Otsuka Pharmaceutical Co. Ltd.

• 大崎 正明

  Laboratories Of Medicinal Chemistry Tokushima Research Institute Otsuka Pharmaceutical Co. Ltd.

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