Sympathomimetic Amines having a 3,4-Dihydrocarbostyril Nucleus

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概要

• 論文の詳細を見る

• A series of new sympathomimetic amines having a 3,4-dihydrocarbostyril nucleus was synthesized. These compounds have two weakly acidic hydrogen atoms in locations similar to those of the hydroxyl groups of adrenergic agents containing catechol. One threo-isomer 1i-threo was synthesized by inversion of the corresponding erythro-isomer by the S_Ni reaction.

• 社団法人日本薬学会の論文
• 1978-05-25

著者

• 楊 永雄

  Tokushima Research Institute, Otsuka Pharmaceutical Co., Ltd.,

• 楊 永雄

  Laboratories of Medicinal Chemistry, Tokushima Research Institute, Otsuka Pharmaceutical Co., Ltd.

• 吉崎 司郎

  (present Address)bio-center Nkk Corporation

• 吉崎 司郎

  Laboratories of Medicinal chemistry, Tokushima Factory, Otsuka Pharmaceutical Co., Ltd.

• 大坪 潤一郎

  Laboratories of Medicinal Chemistry, Tokushima Factory, Otsuka Pharmaceutical Co., Ltd.

• 楊 永雄

  Tokushima Research Institute Otsuka Pharmaceutical Co. Ltd.

• 大坪 潤一郎

  Laboratories Of Medicinal Chemistry Tokushima Factory Otsuka Pharmaceutical Co. Ltd.

関連論文

• 陽性変力作用薬の研究(第3報)6-(Substituted 1-oxoalkyl)-2(1H)quinolinone誘導体の合成
• Studies on Positive Inotropic Agents. II. : Synthesis of(4-Substituted 1-piperazinylcarbonyl)-2-(1H)-quinolinone Derivatives
• Studies on Positive Inotropic Agents. I. Synthesis of 3,4-Dihydro-6-[4-(3,4-dimethoxybenzoyl)-1-piperazinyl]-2 (1H)-quinolinone and Related Compounds
• Synthesis of 5,8-Dihydroxy-3,4-dihydrocarbostyril
• Synthesis and Pharmacological Evaluation of 7-Substituted Procaterol Derivatives
• Synthesis of Procaterol Derivative Having a Piperidylmethanol Group and Its β-Adrenoceptor Stimulant Activities
• Synthesis and Pharmacological Evaluation of Procaterol Derivatives Having a tert-Amino Group
• Studies of the Selective O-Alkylation and Dealkylation of Flavonoids. XII. : A New, Convenient Method for Synthesizing 3,5-Dihydroxy-6,7-dimethoxyflavones from 3,5,6,7-Tetramethoxyflavones
• Synthesis of 5-(2-Allylamino-1-hydroxyalkyl)-8-hydroxycarbostyrils, New β-Adrenoceptor Stimulants
• Synthesis of 8-Hydroxycarbostyril
• Synthesis of 5-(2-Amino-1-hydroxybutyl)-8-hydroxycarbostyril, One of the Major Metabolites of Procaterol
• Oxidation of Procaterol to 5-Formyl-8-hydroxycarbostyril
• Sympathomimetic Amines having a 3,4-Dihydrocarbostyril Nucleus
• Syntheses and β-Adrenergic Blocking Activities of the Optical Isomers of 8-Acetonyloxyl-5-[3-(3,4-dimethoxyphenethylamino)-2-hydroxypropoxy]-3,4-dihydrocarbostyril

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